SCHEMBL20179998

SCHEMBL20179998

COc1cc(CN2CCNCC2)cc(C(F)(F)F)c1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.56
CYP2D6 P10635 4/20 0.56
TSHR P16473 2/20 0.50
TACR1 P25103 3/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
TP53 P04637 1/20 0.48
USP2 O75604 2/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP2C19 P33261 2/20 0.43
CYP2C9 P11712 1/20 0.43
CYP1A2 P05177 1/20 0.42
ADRB1 P08588 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19262510 0.85 CYP2D6 (0.72) CYP3A4CYP2D6TSHRTACR1MEN1
SCHEMBL11628726 0.85 ADRB1 (0.56) MEN1KMT2AALDH1A1CYP1A2ADRB1
SCHEMBL20676125 0.84 CYP2D6 (0.70) CYP3A4CYP2D6TSHRMEN1KMT2A
SCHEMBL28322502 0.81 CYP2D6 (0.48) CYP3A4CYP2D6TSHRMEN1KMT2A
SCHEMBL17320452 0.81 CYP2D6 (0.59) CYP3A4CYP2D6TSHRTACR1MEN1
SCHEMBL19262611 0.80 CYP3A4 (0.61) CYP3A4CYP2D6TSHRTACR1MEN1
SCHEMBL21571720 0.79 MGLL (0.46) CYP3A4CYP2D6TSHRMEN1KMT2A
SCHEMBL28303845 0.78 CYP2D6 (0.59) CYP3A4CYP2D6TSHRMEN1KMT2A
SCHEMBL16907553 0.78 CYP2D6 (0.59) CYP3A4CYP2D6TSHRMEN1KMT2A
SCHEMBL28699525 0.78 CYP3A4 (0.47) CYP3A4CYP2D6TSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018093947-A1 MAGL INHIBITORS ABIDE THERAPEUTICS, INC. (US) 2018-05-24 WO disclosed