SCHEMBL2870543

SCHEMBL2870543

O=C1C=c2c(Nc3c(Cl)cc(F)cc3Cl)nc3ccc(NC(=O)CN4CCOCC4)cc3c2=C[N]1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
GAA P10253 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
ATM Q13315 1/20 0.44
EGFR P00533 4/20 0.43
MAP4K4 O95819 1/20 0.43
ERBB2 P04626 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
POLB P06746 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
KDR P35968 1/20 0.40
ERBB4 Q15303 1/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3501957 0.81 JAK2 (0.53) ALDH1A1GAANPSR1ATMEGFR
SCHEMBL2882063 0.75 TERT (0.36)
SCHEMBL2867747 0.68 JAK2 (0.46) EGFRKDR
SCHEMBL3501684 0.67 JAK2 (0.55) GAAKDM4E
SCHEMBL8110759 0.65 EGFR (0.74) EGFRMAP4K4ERBB2ERBB4
SCHEMBL13597049 0.64 ALDH1A1 (0.77) ALDH1A1GAANPSR1ATML3MBTL1
SCHEMBL11732314 0.64 TERT (0.78) ALDH1A1GAANPSR1ATMPOLB
SCHEMBL13249161 0.64 JAK2 (0.49) GAAKDM4E
SCHEMBL25233242 0.64 ALDH1A1 (0.71) ALDH1A1GAANPSR1ATML3MBTL1
Hydrochloric Acid SCHEMBL11732400 0.63 TERT (0.74) ALDH1A1GAANPSR1ATMPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2200612-A1 INHIBITORS OF JANUS KINASES Merck Sharp & Dohme Corp. (US) 2010-06-30 EP disclosed
WO-2009035575-A1 INHIBITORS OF JANUS KINASES MERCK & CO., INC. (US) 2009-03-19 WO disclosed