SCHEMBL2870569

SCHEMBL2870569

NC(=O)C(N)n1ccc2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.46
SLC6A4 P31645 9/20 0.45
NOTUM Q6P988 1/20 0.44
KMT2A Q03164 1/20 0.42
TSHR P16473 1/20 0.42
RAB9A P51151 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
SLC6A2 P23975 8/20 0.39
NR3C2 P08235 1/20 0.39
CDK4 P11802 1/20 0.37
CCND1 P24385 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14683431 0.81 NOTUM (0.47) LMNASLC6A4NOTUMKMT2ATSHR
SCHEMBL3374081 0.81 NOTUM (0.47) LMNASLC6A4NOTUMKMT2ATSHR
SCHEMBL30641461 0.74 SLC6A2 (0.50) LMNASLC6A4NOTUMKMT2ASLC6A2
SCHEMBL11412911 0.74 KMT2A (0.49) LMNASLC6A4NOTUMKMT2ATSHR
SCHEMBL2976520 0.73 SLC6A4 (0.46) SLC6A4NOTUMSLC6A2CDK4CCND1
SCHEMBL8573980 0.72 SLC6A4 (0.53) SLC6A4NOTUMSLC6A2CDK4CCND1
SCHEMBL2404377 0.72 LMNA (0.41) LMNASLC6A4NOTUMKMT2ATSHR
SCHEMBL30611209 0.72 SLC6A4 (0.44) LMNASLC6A4KMT2ATSHRRAB9A
SCHEMBL10203775 0.71 NOTUM (0.53) SLC6A4NOTUMKMT2ATSHRRAB9A
SCHEMBL526316 0.71 NOTUM (0.49) SLC6A4NOTUMKMT2ATSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383742-B1 SYNTHESIS AND METHODS OF USE OF TETRAHYDROINDOLONE ANALOGUES AND DERIVATIVES SPECTRUM PHARMACEUTICALS INC (US) 2010-10-27 EP disclosed
US-5646300-A NEUROPROTECTIVE AGENTS HOECHST MARION ROUSSEL, INC. (US) 1997-07-08 US disclosed
US-5591866-A NEUROPROTECTIVE AGENTS HOECHST MARION ROUSSEL INC. (US) 1997-01-07 US disclosed
US-5565579-A NEUROPROTECTIVE AGENT HOECHST MARION ROUSSEL INC. (US) 1996-10-15 US disclosed
EP-0563916-B1 (1H-Indol-1-yl)-2-(amino)acetamides and related (1H-indol-1-yl)-(aminoalkyl)amides, intermediates and a process for their preparation and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1995-08-16 EP disclosed
EP-0563916-A1 (1H-Indol-1-yl)-2-(amino)acetamides and related (1H-indol-1-yl)-(aminoalkyl)amides, intermediates and a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-10-06 EP disclosed