SCHEMBL28707172

SCHEMBL28707172

NC(=O)c1csc(Nc2ccc(Cl)cc2)n1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.76
AMY1A P0DUB6 9/20 0.64
TRPC3 Q13507 1/20 0.58
TRPC6 Q9Y210 1/20 0.58
ALDH1A1 P00352 3/20 0.58
MEN1 O00255 3/20 0.58
MAPT P10636 3/20 0.58
KMT2A Q03164 3/20 0.58
NPC1 O15118 2/20 0.58
RAB9A P51151 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
GAA P10253 1/20 0.58
VCP P55072 2/20 0.54
ALOX5 P09917 2/20 0.54
DEGS1 O15121 1/20 0.54
MAP4K4 O95819 1/20 0.54
CYP3A4 P08684 1/20 0.54
ALOX15 P16050 1/20 0.54
TSHR P16473 1/20 0.54
MAPK1 P28482 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL525682 0.88 KDM1A (0.76) KDM1AAMY1ATRPC3TRPC6ALDH1A1
SCHEMBL28717687 0.84 KDM1A (0.67) KDM1AAMY1ATRPC3TRPC6ALDH1A1
SCHEMBL28712067 0.84 KDM1A (0.57) KDM1AAMY1ATRPC3TRPC6MAPT
SCHEMBL27827106 0.84 AMY1A (0.63) KDM1AAMY1AMEN1MAPTKMT2A
SCHEMBL6107121 0.82 KDM1A (0.53) KDM1AAMY1ATRPC3TRPC6MAPT
SCHEMBL29654005 0.82 KDM1A (0.78) KDM1AAMY1AALDH1A1MEN1MAPT
SCHEMBL28707161 0.82 KDM1A (0.78) KDM1AAMY1AALDH1A1MEN1MAPT
SCHEMBL27827048 0.81 AMY1A (0.67) KDM1AAMY1ATRPC3TRPC6MEN1
SCHEMBL5041112 0.79 EGFR (0.73) KDM1AALDH1A1MEN1MAPTKMT2A
SCHEMBL772481 0.78 KDM1A (0.66) KDM1AAMY1ATRPC3TRPC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114249702-B N-aryl- [2,4 '-dithiazole ] -2' -amine compound and preparation and application thereof 沈阳药科大学 2023-09-05 CN disclosed
CN-114249702-A N-aryl- [2,4 '-bithiazole ] -2' -amine compound and preparation and application thereof 沈阳药科大学 2022-03-29 CN disclosed