SCHEMBL772481

SCHEMBL772481

CON(C)C(=O)c1csc(Nc2ccc(Cl)cc2)n1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.66
ALDH1A1 P00352 2/20 0.56
MAPT P10636 5/20 0.54
MAPK1 P28482 1/20 0.54
GFER P55789 1/20 0.54
TRPC3 Q13507 1/20 0.53
TRPC6 Q9Y210 1/20 0.53
AMY1A P0DUB6 7/20 0.53
GAA P10253 3/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
HPGD P15428 1/20 0.52
HTT P42858 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.51
RAB9A P51151 2/20 0.51
NPC1 O15118 1/20 0.51
ALOX5 P09917 1/20 0.48
PKM P14618 1/20 0.48
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL724535 0.89 MAPT (0.69) KDM1AMAPTMAPK1GFERTRPC3
SCHEMBL724563 0.88 MAPT (0.54) KDM1AALDH1A1MAPTMAPK1GFER
SCHEMBL724465 0.87 MAPT (0.54) KDM1AALDH1A1MAPTMAPK1GFER
SCHEMBL723602 0.78 MAPT (0.47) KDM1AMAPTMAPK1GFERGAA
SCHEMBL30621781 0.78 MAPT (0.47) KDM1AMAPTMAPK1GFERGAA
SCHEMBL525682 0.78 KDM1A (0.76) KDM1AALDH1A1MAPTMAPK1TRPC3
SCHEMBL28707172 0.78 KDM1A (0.76) KDM1AALDH1A1MAPTMAPK1TRPC3
SCHEMBL31717584 0.78 RAB9A (0.59) ALDH1A1MAPTGFERGAAMEN1
SCHEMBL5041112 0.76 EGFR (0.73) KDM1AALDH1A1MAPTMAPK1GFER
SCHEMBL16638093 0.76 L3MBTL1 (0.49) ALDH1A1MAPTMAPK1GFERGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250188072-A1 COMPOUNDS FOR TREATMENT OF CANCER UNIVERSITY OF TENNESSEE RESEARCH FOUNDATION (US) 2025-06-12 US disclosed
US-12187720-B2 Compounds for treatment of cancer UNIVERSITY OF TENNESSEE RESEARCH FOUNDATION (US) 2025-01-07 US disclosed
US-11465987-B2 Compounds for treatment of cancer Oncternal Therapeutics, Inc. (US) 2022-10-11 US disclosed
US-20220024912-A1 COMPOUNDS FOR TREATMENT OF CANCER Oncternal Therapeutics, Inc. (US) 2022-01-27 US disclosed
US-11084811-B2 Compounds for treatment of cancer Oncternal Therapeutics, Inc. (US) 2021-08-10 US disclosed
US-20170226086-A1 COMPOUNDS FOR TREATMENT OF CANCER GTx. Inc. (US) 2017-08-10 US disclosed
US-9447049-B2 Compounds for treatment of cancer UNIVERSITY OF TENNESSEE RESEARCH FOUNDATION (US) 2016-09-20 US disclosed
US-8822513-B2 Compounds for treatment of cancer GTX, INC. (US) 2014-09-02 US disclosed
US-20130197049-A1 COMPOUNDS FOR TREATMENT OF CANCER UNIVERSITY OF TENNESSEE RESEARCH FOUNDATION (US) 2013-08-01 US disclosed
US-20120071524-A1 COMPOUNDS FOR TREATMENT OF CANCER ONCTERNAL THERAPEUTICS, INC 2012-03-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12187720-B2 Compounds for treatment of cancer KLK3, BRDT, ACP3 KDM1A 2331/4885ALDH1A1 209/4885MAPT 2614/4885
US-20120071524-A1 COMPOUNDS FOR TREATMENT OF CANCER KLK3, BRDT, ACP3 KDM1A 2331/4885ALDH1A1 209/4885MAPT 2614/4885
US-20130197049-A1 COMPOUNDS FOR TREATMENT OF CANCER KLK3, BRDT, ACP3 KDM1A 2331/4885ALDH1A1 209/4885MAPT 2614/4885
US-11084811-B2 Compounds for treatment of cancer KLK3, BRDT, ACP3 KDM1A 2331/4885ALDH1A1 209/4885MAPT 2614/4885
US-20220024912-A1 COMPOUNDS FOR TREATMENT OF CANCER KLK3, BRDT, ACP3 KDM1A 2331/4885ALDH1A1 209/4885MAPT 2614/4885
US-20170226086-A1 COMPOUNDS FOR TREATMENT OF CANCER KLK3, BRDT, ACP3 KDM1A 2331/4885ALDH1A1 209/4885MAPT 2614/4885
US-20250188072-A1 COMPOUNDS FOR TREATMENT OF CANCER KLK3, BRDT, ACP3 KDM1A 2331/4885ALDH1A1 209/4885MAPT 2614/4885
US-11465987-B2 Compounds for treatment of cancer KLK3, BRDT, ACP3 KDM1A 2331/4885ALDH1A1 209/4885MAPT 2614/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.