SCHEMBL28709229

SCHEMBL28709229

Cc1cc(C)n(-c2cccc(C(CC(=O)O)NC3CCNC3)c2)n1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 6/20 0.44
ITGB6 P18564 6/20 0.44
ITGB8 P26012 6/20 0.44
ITGB5 P18084 5/20 0.44
ITGB1 P05556 5/20 0.44
ITGB3 P05106 4/20 0.44
ITGA5 P08648 1/20 0.44
KCNH2 Q12809 1/20 0.44
SMYD3 Q9H7B4 3/20 0.44
USP7 Q93009 1/20 0.38
CYP26A1 O43174 1/20 0.38
RIPK1 Q13546 2/20 0.37
MAPK14 Q16539 1/20 0.36
KHK P50053 1/20 0.36
KAT6A Q92794 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28709399 0.91 SMYD3 (0.41) ITGAVITGB6ITGB8ITGB5ITGB1
SCHEMBL28698405 0.91 SMYD3 (0.41) ITGAVITGB6ITGB8ITGB5ITGB1
SCHEMBL28709231 0.89 SMYD3 (0.40) ITGAVITGB6ITGB8ITGB5ITGB1
SCHEMBL28709233 0.89 SMYD3 (0.40) ITGAVITGB6ITGB8ITGB5ITGB1
SCHEMBL28699688 0.76 ITGAV (0.39) ITGAVITGB6ITGB8ITGB5ITGB1
SCHEMBL28984876 0.74 KHK (0.38) SMYD3RIPK1KHK
SCHEMBL28692102 0.73 L3MBTL1 (0.45) ITGAVITGB6ITGB8ITGB5ITGB1
SCHEMBL28690085 0.73 CYP26A1 (0.40) ITGAVITGB6ITGB8ITGB5ITGB1
SCHEMBL16115886 0.72 L3MBTL1 (0.45) ITGAVITGB6ITGB8ITGB5ITGB1
SCHEMBL30898093 0.70 ITGAV (0.50) ITGAVITGB6ITGB8ITGB5ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354635-A Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2021-09-07 CN disclosed