SCHEMBL28699688

SCHEMBL28699688

COC(=O)CC(N[C@H]1CCN(C(=O)O)C1)c1cccc(-n2nc(C)cc2C)c1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 5/20 0.39
ITGB5 P18084 5/20 0.39
ITGB6 P18564 5/20 0.39
ITGB8 P26012 5/20 0.39
ITGB3 P05106 4/20 0.39
ITGB1 P05556 4/20 0.39
ITGA5 P08648 1/20 0.39
KCNH2 Q12809 1/20 0.39
RIPK1 Q13546 3/20 0.35
MAPT P10636 2/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
SMYD3 Q9H7B4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28699700 0.89 MAPT (0.41) MAPTKMT2AL3MBTL1MEN1LMNA
SCHEMBL28698405 0.83 SMYD3 (0.41) ITGAVITGB5ITGB6ITGB8ITGB3
SCHEMBL28709399 0.83 SMYD3 (0.41) ITGAVITGB5ITGB6ITGB8ITGB3
SCHEMBL28686054 0.80 WDR5 (0.42) HPGD
SCHEMBL28685987 0.80 ITGAV (0.47) ITGAVITGB5ITGB6ITGB8ITGB3
SCHEMBL28699817 0.80 LMNA (0.41) ITGAVITGB5ITGB6ITGB8ITGB3
SCHEMBL28709233 0.77 SMYD3 (0.40) ITGAVITGB5ITGB6ITGB8ITGB3
SCHEMBL28709231 0.77 SMYD3 (0.40) ITGAVITGB5ITGB6ITGB8ITGB3
SCHEMBL28709229 0.76 ITGAV (0.44) ITGAVITGB5ITGB6ITGB8ITGB3
SCHEMBL24036729 0.76 MAPT (0.42) MAPTHPGDTDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354635-A Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2021-09-07 CN disclosed