SCHEMBL28709784

SCHEMBL28709784

O=C(O)n1cc(-c2cccc([N+](=O)[O-])c2)cn1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.53
F2 P00734 2/20 0.51
PLAU P00749 2/20 0.51
ELANE P08246 2/20 0.51
KLKB1 P03952 1/20 0.51
SMN1; SMN2 Q16637 2/20 0.47
KEAP1 Q14145 3/20 0.46
NFE2L2 Q16236 3/20 0.46
ALDH1A1 P00352 4/20 0.46
MAPT P10636 4/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
PDE4B Q07343 1/20 0.46
TP53 P04637 1/20 0.45
IDO1 P14902 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
PKM P14618 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22353120 0.82 F2 (0.49) TDP1F2PLAUELANEKLKB1
SCHEMBL1019778 0.81 F2 (0.45) TDP1F2PLAUELANEKLKB1
SCHEMBL28712258 0.81 MEN1 (0.44) TDP1F2PLAUELANEKLKB1
SCHEMBL28705422 0.77 EGLN1 (0.50) SMN1; SMN2MAPTNPC1RAB9APDE4B
SCHEMBL28704298 0.77 ELANE (0.47) ELANEMAPTNPC1RAB9AKMT2A
SCHEMBL28710160 0.77 KMO (0.42) NPC1RAB9APDE4BMEN1KMT2A
SCHEMBL2381806 0.75 F2 (0.66) TDP1F2PLAUELANEKLKB1
SCHEMBL6738366 0.74 TSHR (0.76) TDP1SMN1; SMN2ALDH1A1MAPTNPC1
SCHEMBL28709782 0.73 GRM5 (0.52) IDO1
SCHEMBL29526232 0.73 TSHR (0.67) TDP1SMN1; SMN2NFE2L2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114057646-A Pyrazole derivative and application thereof in preparation of antitumor drugs 常州大学 2022-02-18 CN disclosed