SCHEMBL28713751

SCHEMBL28713751

COc1ccc(-c2cnn(C(=O)O)c2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 1/20 0.53
EGLN1 Q9GZT9 1/20 0.50
KDR P35968 3/20 0.45
MAP4K4 O95819 2/20 0.44
PLK4 O00444 1/20 0.44
AURKA O14965 1/20 0.44
DYRK3 O43781 1/20 0.44
NTRK1 P04629 1/20 0.44
INSR P06213 1/20 0.44
CDK1 P06493 1/20 0.44
FGFR1 P11362 1/20 0.44
FLT1 P17948 1/20 0.44
CDK2 P24941 1/20 0.44
MARK3 P27448 1/20 0.44
FLT4 P35916 1/20 0.44
FLT3 P36888 1/20 0.44
CLK2 P49760 1/20 0.44
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
IRAK1 P51617 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28712249 0.81 F2 (0.45) EGLN1KDRMAP4K4MKNK2ALDH1A1
SCHEMBL29010236 0.79 PARP1 (0.48) MAPKAPK2EGLN1KDRALDH1A1ATM
SCHEMBL28700571 0.78 MAP4K4 (0.50) EGLN1MAP4K4ALDH1A1KDM4EMAPT
SCHEMBL28710155 0.78 BCL2L1 (0.46) EGLN1KDRMAP4K4ALDH1A1KDM4E
SCHEMBL3076935 0.78 KCNH2 (0.39) ALDH1A1KDM4ESMN1; SMN2
SCHEMBL5646211 0.76 MAPKAPK2 (0.51) MAPKAPK2EGLN1KDRMAP4K4PLK4
SCHEMBL28705426 0.75 MMP3 (0.44) EGLN1MAP4K4FLT1HDAC2
SCHEMBL5990507 0.74 CLK1 (0.51) MAPKAPK2KDRMAP4K4PLK4AURKA
SCHEMBL182164 0.74 MAPKAPK2 (0.79) MAPKAPK2EGLN1MAP4K4ALDH1A1KDM4E
SCHEMBL13763422 0.73 GAA (0.47) MAPKAPK2KDRMAP4K4PLK4AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114057646-A Pyrazole derivative and application thereof in preparation of antitumor drugs 常州大学 2022-02-18 CN disclosed