SCHEMBL28717337

SCHEMBL28717337

COc1cc(-n2cc(-c3ccc4nc(N)[nH]c(=O)c4c3)nn2)cc(OC)c1OC

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SQSTM1 Q13501 1/20 0.69
RNF168 Q8IYW5 1/20 0.46
DHFR P00374 1/20 0.44
STIM1 Q13586 5/20 0.43
ORAI1 Q96D31 5/20 0.43
KATNA1 O75449 1/20 0.41
CYP1B1 Q16678 1/20 0.40
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
TYMS P04818 1/20 0.38
ROCK2 O75116 2/20 0.37
PDGFRB P09619 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA5A P35218 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28707826 0.89 SQSTM1 (0.64) SQSTM1RNF168STIM1ORAI1KATNA1
SCHEMBL28714921 0.82 SQSTM1 (1.00) SQSTM1RNF168DHFRSTIM1ORAI1
SCHEMBL4755097 0.70 TYMS (0.44) DHFRKMT2AKDM4EMEN1ALDH1A1
SCHEMBL19126482 0.70 SQSTM1 (0.45) SQSTM1STIM1ORAI1CYP1B1KDM4E
SCHEMBL28704210 0.70 SQSTM1 (0.78) SQSTM1DHFRSTIM1ORAI1CYP1B1
SCHEMBL28713001 0.67 SQSTM1 (0.73) SQSTM1DHFRSTIM1ORAI1CYP1B1
SCHEMBL28721769 0.67 SQSTM1 (0.74) SQSTM1DHFRSTIM1ORAI1CYP1B1
SCHEMBL14072478 0.67 KDM4E (0.56) KMT2AKDM4EMEN1ALDH1A1POLB
SCHEMBL20393728 0.67 SQSTM1 (0.51) SQSTM1CYP1B1KDM4EALDH1A1MAPT
SCHEMBL12497434 0.66 CYP1B1 (0.55) SQSTM1STIM1ORAI1CYP1B1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114230557-B Quinazoline-substituted 1,2,3-triazole derivative, and pharmaceutical composition, preparation method and application thereof 深圳大学 2023-01-06 CN disclosed
CN-114230557-A Quinazoline-substituted 1,2, 3-triazole derivative, and pharmaceutical composition, preparation method and application thereof 深圳大学 2022-03-25 CN disclosed