SCHEMBL287196

SCHEMBL287196

COc1ccc(C2C=NC=C(C(=O)N(CC(=O)c3cccs3)NS(C)(=O)=O)C2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.41
ALDH1A1 P00352 4/20 0.38
NPSR1 Q6W5P4 3/20 0.38
HPGD P15428 3/20 0.38
KDM4E B2RXH2 1/20 0.38
ADRB2 P07550 1/20 0.38
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
POLB P06746 2/20 0.38
MAPT P10636 5/20 0.37
RAB9A P51151 4/20 0.37
GAA P10253 3/20 0.37
LMNA P02545 3/20 0.37
HTT P42858 1/20 0.37
PKM P14618 1/20 0.36
NPC1 O15118 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TP53 P04637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MAPK1 P28482 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL287518 0.75 ALDH1A1 (0.35) ALDH1A1NPSR1HPGDMEN1KMT2A
SCHEMBL288004 0.74 ALDH1A1 (0.48) ALDH1A1NPSR1HPGDMEN1KMT2A
SCHEMBL287418 0.71 ALDH1A1 (0.35) ALDH1A1HPGDMEN1KMT2APOLB
SCHEMBL287275 0.71 GSK3B (0.36) ALDH1A1NPSR1HPGDMEN1KMT2A
SCHEMBL287292 0.70 ALDH1A1 (0.34) ALDH1A1HPGDMEN1KMT2APOLB
SCHEMBL288036 0.68 POLB (0.39) HSD17B10ALDH1A1MEN1KMT2APOLB
SCHEMBL286928 0.66 ALDH1A1 (0.34) ALDH1A1HPGDMEN1KMT2APOLB
SCHEMBL287274 0.65 ALDH1A1 (0.33) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL287118 0.65 KMT2A (0.33) ALDH1A1NPSR1HPGDKDM4EMEN1
SCHEMBL286738 0.65 KMT2A (0.38) ALDH1A1HPGDMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427432-A2 NOVEL HETEROCYCLIC COMPOUNDS Torrent Pharmaceuticals Limited (IN) 2012-03-14 EP claimed
WO-2010128528-A2 NOVEL HETEROCYCLIC COMPOUNDS TORRENT PHARMACEUTICALS LIMITED (IN) 2010-11-11 WO claimed