SCHEMBL28720392

SCHEMBL28720392

O=C(OC(C#Cc1ccccc1)c1ccccn1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
TSHR P16473 1/20 0.41
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
MITF O75030 1/20 0.39
PKM P14618 1/20 0.39
CDK5 Q00535 1/20 0.39
CDK5R1 Q15078 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 1/20 0.38
KMT2A Q03164 4/20 0.37
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ALDH1A1 P00352 1/20 0.37
KDM4E B2RXH2 1/20 0.36
LMNA P02545 2/20 0.36
METAP2 P50579 1/20 0.36
METAP1 P53582 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28714044 0.86 TSHR (0.44) TSHRCYP1A2CYP3A4KMT2AMEN1
SCHEMBL9738786 0.83 KMT2A (0.48) TP53TSHRNPC1RAB9AMITF
SCHEMBL28354626 0.79 TSHR (0.49) TP53TSHRNPC1RAB9ANCOA3
SCHEMBL28717072 0.77 ALDH1A1 (0.44) TSHRNPC1RAB9ACYP1A2CYP3A4
SCHEMBL28719226 0.76 ALDH1A1 (0.51) TSHRNPC1RAB9ACYP1A2CYP3A4
SCHEMBL28717041 0.76 TSHR (0.52) TSHRNPC1RAB9APKMCDK5
SCHEMBL28712253 0.74 ALDH1A1 (0.43) TSHRCYP3A4ALDH1A1KDM4ELMNA
SCHEMBL13719456 0.73 TSHR (0.49) TP53TSHRNPC1RAB9ACYP1A2
SCHEMBL29092696 0.68 NPC1 (0.43) TP53NPC1RAB9APKMCYP1A2
SCHEMBL11179575 0.67 SMN1; SMN2 (0.52) TSHRCYP1A2CYP3A4KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116903612-A Diaryl methane derivative containing indolizine and preparation method and application thereof 江西师范大学 2023-10-20 CN disclosed
CN-115650980-A Oxindole compound and preparation method and application thereof 江西师范大学 2023-01-31 CN disclosed
CN-114163436-A Diarylmethane derivative containing indolizine and preparation method and application thereof 江西师范大学 2022-03-11 CN disclosed
CN-114105978-A Oxindole compound and preparation method and application thereof 江西师范大学 2022-03-01 CN disclosed