SCHEMBL2872122

SCHEMBL2872122

CC(C)Oc1cc2c(cc1C13CC4CC(CC(C4)C1)C3)CN(CC(N)(CO)CO)CC2.CCCCCCCCOc1ccc(CCC(N)(CO)CO)cc1C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 11/20 0.44
S1PR3 Q99500 3/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C8 P10632 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
PPARG P37231 1/20 0.34
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34
TNNC1 P63316 6/20 0.34
S1PR4 O95977 2/20 0.34
S1PR5 Q9H228 2/20 0.34
SGPL1 O95470 1/20 0.34
GPR183 P32249 1/20 0.34
CERS2 Q96G23 1/20 0.34
SPHK2 Q9NRA0 2/20 0.33
SPHK1 Q9NYA1 1/20 0.33
S1PR2 O95136 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL566500 0.84 S1PR1 (0.35) S1PR1S1PR3
SCHEMBL566429 0.82 S1PR1 (0.60) S1PR1S1PR3CYP3A4CYP2C8CYP2D6
Hydrochloric Acid SCHEMBL567052 0.81 S1PR1 (0.59) S1PR1S1PR3CYP3A4CYP2C8CYP2D6
SCHEMBL10139272 0.77 S1PR1 (0.39) S1PR1S1PR3CYP3A4CYP2C8CYP2D6
Hydrochloric Acid SCHEMBL566087 0.76 S1PR1 (0.39) S1PR1S1PR3CYP3A4CYP2C8CYP2D6
SCHEMBL822473 0.74
SCHEMBL10171069 0.73 S1PR1 (0.57) S1PR1S1PR3CYP3A4CYP2C8CYP2D6
SCHEMBL565912 0.70 S1PR1 (0.83) S1PR1S1PR3CYP3A4CYP2C8CYP2D6
SCHEMBL10139273 0.69 S1PR1 (0.43) S1PR1S1PR3CYP3A4CYP2C8CYP2D6
SCHEMBL566953 0.68 HDAC11 (0.33) S1PR1CYP3A4CYP2D6PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010042998-A1 S1P RECEPTORS MODULATORS AKAAL PHARMA PTY LTD (AU) 2010-04-22 WO claimed