SCHEMBL2872141

SCHEMBL2872141

CC(C)(C)OC(=O)NCCCNC(=O)C1(C(=O)O)C=CNC(c2ccccn2)=C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 3/20 0.38
PDPK1 O15530 1/20 0.38
CCNB2 O95067 1/20 0.38
PRKCB P05771 1/20 0.38
CDK1 P06493 1/20 0.38
LYN P07948 1/20 0.38
CCNB1 P14635 1/20 0.38
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38
GSK3B P49841 1/20 0.38
RPS6KA3 P51812 1/20 0.38
CCNA1 P78396 1/20 0.38
CCNB3 Q8WWL7 1/20 0.38
BCHE P06276 1/20 0.37
ACACB O00763 1/20 0.37
ACACA Q13085 1/20 0.37
NPSR1 Q6W5P4 2/20 0.36
MALT1 Q9UDY8 1/20 0.36
BRD4 O60885 1/20 0.36
AKT1 P31749 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2871839 0.96 BCHE (0.40) ATMPDPK1CCNB2PRKCBCDK1
SCHEMBL2875247 0.84 METAP1 (0.34) ACACBACACACYP3A4
SCHEMBL2876748 0.83 ASAH1 (0.41) L3MBTL1KDM4E
SCHEMBL2878070 0.78 HPGDS (0.46) CYP3A4KDM4E
SCHEMBL93597 0.76 KDM4E (0.42) L3MBTL1KDM4ETDP1
Thiocyanic Acid SCHEMBL1615957 0.70 KDM4E (0.37) L3MBTL1KDM4E
SCHEMBL6300342 0.68 STK17B (0.52) BCHEMALT1BRD4STK17BSTK17A
SCHEMBL8357911 0.67 KDM4E (0.40) L3MBTL1KDM4E
SCHEMBL4422174 0.67 AKT1 (0.53) ACACBACACAAKT1CKS1BSKP1
SCHEMBL30453099 0.67 AKT1 (0.53) ACACBACACAAKT1CKS1BSKP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010043866-A2 HISTONE LYSINE DEMETHYLASE INHIBITORS ISIS INNOVATION LIMITED (GB) 2010-04-22 WO disclosed