SCHEMBL28723331

SCHEMBL28723331

C#CCCS(=O)(=O)N1CCC(OC(N)=O)CC1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.36
MAPT P10636 3/20 0.35
POLB P06746 1/20 0.35
ALDH1A1 P00352 6/20 0.35
LMNA P02545 4/20 0.35
BCHE P06276 2/20 0.35
CCND1 P24385 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
CDK6 Q00534 1/20 0.34
EPHX2 P34913 1/20 0.34
KDM4E B2RXH2 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
ALOX15 P16050 1/20 0.32
MMP1 P03956 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29077481 0.78 EPHX2 (0.40) NPC1MAPTPOLBALDH1A1LMNA
SCHEMBL29172800 0.77 SMYD3 (0.42) NPC1ALDH1A1LMNAKDM4EHTT
SCHEMBL19863561 0.77 CCND1 (0.38) NPC1MAPTALDH1A1LMNACCND1
SCHEMBL29260039 0.74 BCHE (0.42) BCHESMN1; SMN2
SCHEMBL19857411 0.74 ALDH1A1 (0.37) NPC1MAPTALDH1A1LMNACCND1
SCHEMBL29077624 0.73 ATM (0.39) MAPTPOLBALDH1A1LMNASMN1; SMN2
SCHEMBL19857361 0.72 TSHR (0.47) NPC1MAPTALDH1A1CCND1CCNE1
SCHEMBL28670500 0.72 BCHE (0.60) BCHESMN1; SMN2
SCHEMBL29191942 0.72 EPHX2 (0.41) POLBEPHX2SMN1; SMN2
SCHEMBL28759274 0.72 TP53 (0.51) MAPTALDH1A1LMNAKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114394966-A Pyridopyrimidinone CDK2/4/6 inhibitors 辉瑞公司 2022-04-26 CN disclosed