SCHEMBL28725071

SCHEMBL28725071

CC(C)c1noc(N2CCC(C[O])CC2)n1

nearest known ligand 0.67

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 18/20 0.67
GPR183 P32249 1/20 0.48
CNR2 P34972 1/20 0.38
KCNH2 Q12809 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11956913 0.87 GPR119 (0.68) GPR119GPR183CNR2KCNH2LMNA
SCHEMBL6118208 0.85 GPR119 (0.67) GPR119GPR183CNR2KCNH2LMNA
SCHEMBL387876 0.85 GPR119 (0.71) GPR119GPR183CNR2KCNH2LMNA
SCHEMBL5779093 0.84 GPR119 (0.74) GPR119GPR183CNR2LMNAMAPT
SCHEMBL19450515 0.84 GPR119 (0.65) GPR119GPR183CNR2KCNH2
SCHEMBL1922450 0.84 GPR119 (0.65) GPR119GPR183CNR2KCNH2
SCHEMBL22514057 0.83 GPR119 (0.63) GPR119GPR183CNR2KCNH2LMNA
SCHEMBL19454550 0.83 GPR119 (0.68) GPR119GPR183CNR2KCNH2
SCHEMBL18843833 0.83 GPR119 (0.63) GPR119GPR183CNR2KCNH2LMNA
SCHEMBL21665285 0.82 GPR119 (0.62) GPR119GPR183CNR2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109415381-B Thiazolopyridine derivatives as GPR119 agonists 人类制药有限公司 2022-03-25 CN disclosed