SCHEMBL28736331

SCHEMBL28736331

COc1ccc(C2=NN(C(=O)OCc3ccccc3)C(c3cc(OC)c(OC)c(OC)c3)C2)cc1

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.57
RAB9A P51151 1/20 0.57
MAOA P21397 3/20 0.56
MAOB P27338 1/20 0.53
ABCB1 P08183 3/20 0.53
ABCG2 Q9UNQ0 3/20 0.53
CA1 P00915 2/20 0.52
CA2 P00918 2/20 0.52
KDM4E B2RXH2 1/20 0.52
ALDH1A1 P00352 1/20 0.52
HPGD P15428 1/20 0.52
MEN1 O00255 1/20 0.52
HTT P42858 1/20 0.52
KMT2A Q03164 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28736370 0.94 MAOB (0.58) MAOAMAOBABCB1ABCG2CA1
SCHEMBL28736252 0.91 MAOA (0.54) MAOAMAOBABCB1ABCG2KMT2A
SCHEMBL28736399 0.88 MAOA (0.62) NPC1RAB9AMAOAMAOBCA1
SCHEMBL28736320 0.88 MAOA (0.58) MAOAMAOBABCB1ABCG2CA1
SCHEMBL28736288 0.86 CA1 (0.55) NPC1RAB9AMAOACA1CA2
SCHEMBL28736360 0.85 MAOA (0.68) RAB9AMAOAMAOBABCB1ABCG2
SCHEMBL28260637 0.85 CA1 (0.61) NPC1RAB9AMAOAMAOBABCB1
SCHEMBL28260652 0.84 CA1 (0.62) NPC1RAB9AMAOAMAOBABCB1
SCHEMBL28736474 0.83 MAOA (0.60) MAOAMAOBABCB1ABCG2CA1
SCHEMBL23052465 0.82 NPC1 (0.71) NPC1RAB9AMAOAMAOBABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109020888-B Pyrazoline structure-containing microtubule polymerization inhibitor and application thereof 南京大学 2021-11-16 CN claimed
CN-109020888-B Pyrazoline structure-containing microtubule polymerization inhibitor and application thereof 南京大学 2021-11-16 CN disclosed