SCHEMBL28260652

SCHEMBL28260652

COc1ccc(C2=NN(C(=O)O)C(c3cc(OC)c(OC)c(OC)c3)C2)cc1

nearest known ligand 0.71

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.62
CA2 P00918 4/20 0.62
NPC1 O15118 1/20 0.61
RAB9A P51151 1/20 0.61
MAOA P21397 2/20 0.57
MAOB P27338 2/20 0.57
ABCB1 P08183 3/20 0.56
ABCG2 Q9UNQ0 3/20 0.56
PTGS2 P35354 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23052167 0.91 NPC1 (0.71) NPC1RAB9AMAOAMAOBABCB1
SCHEMBL23052465 0.91 NPC1 (0.71) NPC1RAB9AMAOAMAOBABCB1
SCHEMBL28260640 0.91 MAOB (0.67) CA1CA2MAOAMAOBABCB1
SCHEMBL28260637 0.90 CA1 (0.61) CA1CA2NPC1RAB9AMAOA
SCHEMBL28258967 0.89 CA1 (0.59) CA1CA2MAOAMAOBABCB1
SCHEMBL28260653 0.89 CA1 (0.71) CA1CA2MAOAMAOBABCB1
SCHEMBL28260648 0.88 PTGS2 (0.58) CA1CA2MAOAMAOBABCB1
SCHEMBL28736399 0.87 MAOA (0.62) CA1CA2NPC1RAB9AMAOA
SCHEMBL28736288 0.84 CA1 (0.55) CA1CA2NPC1RAB9AMAOA
SCHEMBL28736331 0.84 NPC1 (0.57) CA1CA2NPC1RAB9AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109020888-A A kind of microtubule polymerization inhibitor of the structure containing pyrazoline and its application 南京大学 2018-12-18 CN claimed
CN-109020888-A A kind of microtubule polymerization inhibitor of the structure containing pyrazoline and its application 南京大学 2018-12-18 CN disclosed