SCHEMBL28743751

SCHEMBL28743751

COc1ccc(-c2cncnc2)c(OC)c1OC

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.53
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
EGFR P00533 1/20 0.44
KDR P35968 1/20 0.44
ADORA1 P30542 1/20 0.42
CYP17A1 P05093 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
HDAC4 P56524 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
AMY1A P0DUB6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27503313 0.81 CYP17A1 (0.60) KDM4EMAPK1HTTSMN1; SMN2HSD17B10
SCHEMBL13804249 0.78 ERN1 (0.47) ERN1EGFRKDRCYP17A1CYP11B1
SCHEMBL642228 0.77 HDAC4 (0.58) ERN1KDM4EALDH1A1LMNAMAPT
SCHEMBL29788008 0.75 HDAC4 (0.53) ERN1KDM4EALDH1A1LMNAMAPT
SCHEMBL4579619 0.75 HDAC4 (0.53) ERN1KDM4EALDH1A1LMNAMAPT
SCHEMBL6754272 0.73 CYP1A2 (0.54) ERN1KDM4EALDH1A1LMNAHPGD
SCHEMBL8502557 0.73 CYP17A1 (0.55) ERN1KDM4EALDH1A1LMNAMAPT
SCHEMBL3674074 0.72 CA9 (0.50) KDM4EALDH1A1MAPTHPGDSMN1; SMN2
SCHEMBL30701949 0.72 CA9 (0.50) KDM4EALDH1A1MAPTHPGDSMN1; SMN2
SCHEMBL7260001 0.72 ERN1 (0.49) ERN1KDM4EALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100491352-C Asymmetrical cyclic diamine compound KOWA CO (JP) 2009-05-27 CN disclosed
CN-1242992-C Cyclic diamine compounds bearing six-membered cyclic groups KOWA CO (JP) 2006-02-22 CN disclosed
CN-1520402-A Unsymmetrical cyclic diamine compound ������������ʽ���� 2004-08-11 CN disclosed
CN-1520400-A Cyclic diamine compounds with six-membered cyclic groups ������������ʽ���� 2004-08-11 CN disclosed
CN-1438890-A Adenosine receptor modulators HOFFMANNLA ROCHE AG F (CH) 2003-08-27 CN disclosed