SCHEMBL28748558

SCHEMBL28748558

CN(C)C/C(=C(\C=O)c1ccc(F)cc1)c1ccnc(Cl)n1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.33
GRM5 P41594 2/20 0.31
CYP1A2 P05177 3/20 0.31
CYP3A4 P08684 2/20 0.31
CYP2C19 P33261 2/20 0.31
USP2 O75604 1/20 0.31
CYP2D6 P10635 1/20 0.31
ABL1 P00519 1/20 0.31
BCR P11274 1/20 0.31
KMT2A Q03164 3/20 0.31
MEN1 O00255 1/20 0.30
MAPK11 Q15759 1/20 0.30
MAPK14 Q16539 1/20 0.30
GRM1 Q13255 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27516993 1.00 TRPV1 (0.33) TRPV1GRM5CYP1A2CYP3A4CYP2C19
SCHEMBL27637673 0.84 ALDH1A1 (0.36) CYP1A2CYP3A4CYP2C19USP2MAPK14
SCHEMBL27337618 0.76 LTA4H (0.45) CYP1A2CYP2C19KMT2AGRM1
SCHEMBL27523731 0.76 LTA4H (0.45) CYP1A2CYP2C19KMT2AGRM1
SCHEMBL5261066 0.70 CYP1A2 (0.38) TRPV1GRM5CYP1A2CYP3A4CYP2C19
SCHEMBL5261054 0.70 CYP1A2 (0.38) TRPV1GRM5CYP1A2CYP3A4CYP2C19
SCHEMBL22594425 0.70 LTA4H (0.49) TRPV1GRM5ABL1BCRKMT2A
SCHEMBL27555390 0.69 BCL2L1 (0.37) CYP1A2CYP2C19KMT2AGRM1
SCHEMBL5788690 0.66 LTA4H (0.49) CYP1A2CYP2C19USP2KMT2AMEN1
SCHEMBL27608096 0.66 NAPRT (0.42) USP2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1342157-A Substituted pyrazoles ASP38 kinase inhibitors SEARLE & CO (US) 2002-03-27 CN disclosed