SCHEMBL28749916

SCHEMBL28749916

Cn1c(=O)c2c(ncn2CCc2ccccc2)n(CCO)c1=O

nearest known ligand 0.73

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.73
PDE4A P27815 3/20 0.66
PDE4B Q07343 3/20 0.66
PDE4C Q08493 3/20 0.66
PDE4D Q08499 3/20 0.66
CNOT7 Q9UIV1 11/20 0.65
TSHR P16473 1/20 0.63
POLB P06746 1/20 0.61
HIF1A Q16665 1/20 0.61
PARN O95453 1/20 0.61
ADORA2B P29275 3/20 0.59
LMNA P02545 1/20 0.59
PDE1A P54750 1/20 0.58
PDE1B Q01064 1/20 0.58
PDE1C Q14123 1/20 0.58
ADORA2A P29274 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
RXFP1 Q9HBX9 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL555404 0.89 PDE1A (0.73) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL27583105 0.88 CNOT7 (0.78) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL28752105 0.86 CNOT7 (0.80) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL17786242 0.85 ALDH1A1 (1.00) ALDH1A1CNOT7TSHRPOLBHIF1A
SCHEMBL27600238 0.85 ALDH1A1 (0.72) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL27600252 0.83 ALDH1A1 (0.66) ALDH1A1CNOT7TSHRPOLBHIF1A
SCHEMBL27583005 0.83 ALDH1A1 (0.69) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL27600280 0.81 CNOT7 (0.80) ALDH1A1CNOT7TSHRPOLBHIF1A
SCHEMBL28752095 0.80 ALDH1A1 (0.75) ALDH1A1CNOT7TSHRPOLBHIF1A
SCHEMBL27582971 0.80 KDM4E (0.62) ALDH1A1PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101293888-B Xanthine derivative, production and use thereof as a medicament BOEHRINGER INGELHEIM PHARMA 2013-09-25 CN disclosed
CN-101293888-A Xanthine derivative, production and use thereof as a medicament BOEHRINGER INGELHEIM PHARMA (DE) 2008-10-29 CN disclosed
CN-100408579-C Xanthine derivatives, process for their preparation and their use as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA (DE) 2008-08-06 CN disclosed
CN-1492870-A Xanthine derivatives, process for their preparation and their use as pharmaceutical compositions ���ָ��Ӣ��ķ�������Ϲ�˾ 2004-04-28 CN disclosed