SCHEMBL28752105

SCHEMBL28752105

CCCCCCn1c(=O)n(C)c(=O)c2c1ncn2CCc1ccccc1

nearest known ligand 0.80

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNOT7 Q9UIV1 10/20 0.80
ALDH1A1 P00352 1/20 0.70
ADORA2A P29274 3/20 0.65
TSHR P16473 1/20 0.64
PDE4A P27815 4/20 0.62
PDE4B Q07343 4/20 0.62
PDE4C Q08493 4/20 0.62
PDE4D Q08499 4/20 0.62
ADORA2B P29275 2/20 0.62
PARN O95453 1/20 0.61
POLB P06746 1/20 0.58
HIF1A Q16665 1/20 0.58
PDE1A P54750 1/20 0.56
PDE1B Q01064 1/20 0.56
PDE1C Q14123 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL556098 0.90 PDE1A (0.70) CNOT7ALDH1A1ADORA2ATSHRPDE4A
SCHEMBL27583105 0.88 CNOT7 (0.78) CNOT7ALDH1A1ADORA2ATSHRPDE4A
SCHEMBL28749916 0.86 ALDH1A1 (0.73) CNOT7ALDH1A1ADORA2ATSHRPDE4A
SCHEMBL27600284 0.83 ALDH1A1 (0.70) CNOT7ALDH1A1ADORA2APDE4APDE4B
SCHEMBL17786242 0.83 ALDH1A1 (1.00) CNOT7ALDH1A1TSHRADORA2BPOLB
SCHEMBL27600238 0.83 ALDH1A1 (0.72) CNOT7ALDH1A1ADORA2ATSHRPDE4A
SCHEMBL27600280 0.82 CNOT7 (0.80) CNOT7ALDH1A1TSHRPARNPOLB
SCHEMBL27583005 0.81 ALDH1A1 (0.69) CNOT7ALDH1A1ADORA2ATSHRPDE4A
SCHEMBL27583016 0.80 CYP1A2 (0.58) CNOT7ALDH1A1TSHR
SCHEMBL3112709 0.80 POLB (0.68) CNOT7ALDH1A1ADORA2ATSHRPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101293888-B Xanthine derivative, production and use thereof as a medicament BOEHRINGER INGELHEIM PHARMA 2013-09-25 CN disclosed
CN-101293888-A Xanthine derivative, production and use thereof as a medicament BOEHRINGER INGELHEIM PHARMA (DE) 2008-10-29 CN disclosed
CN-100408579-C Xanthine derivatives, process for their preparation and their use as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA (DE) 2008-08-06 CN disclosed
CN-1492870-A Xanthine derivatives, process for their preparation and their use as pharmaceutical compositions ���ָ��Ӣ��ķ�������Ϲ�˾ 2004-04-28 CN disclosed