SCHEMBL2875012

SCHEMBL2875012

Cc1cc(Cl)c(COc2ccc3nc(C)cc(-c4n[nH]cc4CO)c3c2)c(Cn2cccc(C#N)c2=O)n1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 4/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C19 P33261 1/20 0.34
PKM P14618 1/20 0.32
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
MRGPRX4 Q96LA9 2/20 0.31
ADAM17 P78536 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2868557 0.92 CYP3A4 (0.33) BDKRB2CYP3A4CYP2C19MRGPRX4
SCHEMBL1564368 0.87 BDKRB2 (0.47) BDKRB2CYP3A4CYP2C19
SCHEMBL2877771 0.87 BDKRB2 (0.34) BDKRB2CYP3A4CYP2C19MRGPRX4
SCHEMBL2872758 0.85 BDKRB2 (0.46) BDKRB2CYP3A4CYP2C19MRGPRX4
SCHEMBL2878108 0.83 BDKRB2 (0.45) BDKRB2CYP3A4CYP2C19
SCHEMBL2878084 0.82 BDKRB2 (0.34) BDKRB2CYP3A4CYP2C19
SCHEMBL2877380 0.82 BDKRB2 (0.40) BDKRB2CYP3A4CYP2C19
SCHEMBL2877603 0.82 BDKRB2 (0.40) BDKRB2CYP3A4CYP2C19
SCHEMBL2876863 0.80 BDKRB2 (0.49) BDKRB2CYP3A4CYP2C19
SCHEMBL13146270 0.80 BDKRB2 (0.48) BDKRB2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2144897-B1 8-OXY-QUINOLINE DERIVATIVES AS BRADYKININ B2 RECEPTOR MODULATORS JERINI AG (DE) 2010-10-20 EP claimed