SCHEMBL28752123

SCHEMBL28752123

Cn1c(=O)c2c(nc(Cl)n2CCc2ccccc2)n(CC2CC2)c1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.54
PDE4A P27815 2/20 0.54
PDE4B Q07343 2/20 0.54
PDE4C Q08493 2/20 0.54
PDE4D Q08499 2/20 0.54
TSHR P16473 10/20 0.53
LMNA P02545 3/20 0.53
ADORA3 P0DMS8 1/20 0.52
GAA P10253 1/20 0.48
ALDH1A1 P00352 5/20 0.48
TP53 P04637 1/20 0.48
ALOX15 P16050 1/20 0.48
MAPK1 P28482 3/20 0.48
HSD17B10 Q99714 1/20 0.48
HTT P42858 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
RECQL P46063 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HPGD P15428 1/20 0.47
KDM4E B2RXH2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL555649 0.91 PDE5A (0.62) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL555312 0.90 ALDH1A1 (0.55) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL27600589 0.89 LMNA (0.62) TSHRLMNAALDH1A1TP53ALOX15
SCHEMBL27600387 0.85 LMNA (0.58) TSHRLMNAALDH1A1MAPK1HSD17B10
SCHEMBL27582891 0.84 LMNA (0.57) TSHRLMNAADORA3ALDH1A1MAPK1
SCHEMBL555395 0.84 HTT (0.60) TSHRLMNAALDH1A1TP53ALOX15
SCHEMBL27582885 0.84 LMNA (0.73) TSHRLMNAALDH1A1TP53ALOX15
SCHEMBL27600370 0.83 LMNA (0.57) TSHRLMNAALDH1A1TP53ALOX15
SCHEMBL28749937 0.82 LMNA (0.55) TSHRLMNAALDH1A1TP53ALOX15
SCHEMBL28749929 0.81 HIF1A (0.62) TSHRLMNAADORA3GAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101293888-B Xanthine derivative, production and use thereof as a medicament BOEHRINGER INGELHEIM PHARMA 2013-09-25 CN disclosed
CN-101293888-A Xanthine derivative, production and use thereof as a medicament BOEHRINGER INGELHEIM PHARMA (DE) 2008-10-29 CN disclosed
CN-100408579-C Xanthine derivatives, process for their preparation and their use as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA (DE) 2008-08-06 CN disclosed
CN-1492870-A Xanthine derivatives, process for their preparation and their use as pharmaceutical compositions ���ָ��Ӣ��ķ�������Ϲ�˾ 2004-04-28 CN disclosed