SCHEMBL2875358

SCHEMBL2875358

CCCCc1ccc(C#Cc2ccc(CN(Cc3cccc4c3OC(C)(C)OC4=O)C(=O)CCC3CCCC3)cc2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.37
HTR5A P47898 7/20 0.36
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
HTR1D P28221 1/20 0.35
HTR1B P28222 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR7 P34969 1/20 0.35
ADRA1B P35368 1/20 0.35
DRD3 P35462 1/20 0.35
HTR2B P41595 1/20 0.35
HTR6 P50406 1/20 0.35
POLB P06746 1/20 0.35
CNR2 P34972 1/20 0.35
ALDH1A1 P00352 2/20 0.34
LTB4R2 Q9NPC1 3/20 0.33
MMP2 P08253 1/20 0.32
MMP9 P14780 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2859640 0.86 SLC6A4 (0.38) SLC6A4HTR5AHTR1ADRD2DRD4
SCHEMBL2855107 0.81 PTPN11 (0.36) SLC6A4HTR5AHTR1ADRD2DRD4
SCHEMBL2858908 0.81 PTPN11 (0.36) SLC6A4HTR5AHTR1ADRD2DRD4
SCHEMBL13513480 0.78 SLC6A4 (0.45) SLC6A4HTR5AHTR1ADRD2DRD4
SCHEMBL1734729 0.77 RARB (0.46) SLC6A4HTR5AHTR1ADRD2DRD4
SCHEMBL4457062 0.76 SLC6A4 (0.35) SLC6A4HTR5AHTR1ADRD2DRD4
SCHEMBL2868663 0.76 LTB4R2 (0.34) SLC6A4HTR5AHTR1ADRD2DRD4
SCHEMBL2875007 0.74 SLC6A4 (0.43) SLC6A4HTR5AHTR1ADRD2DRD4
SCHEMBL2859740 0.74 HTR5A (0.35) SLC6A4HTR5ACNR2LTB4R2PTPN11
SCHEMBL2853646 0.73 PTPN11 (0.39) POLBALDH1A1LTB4R2MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654247-B1 ALKYNYL ARYL CARBOXAMIDES MERCK SERONO SA (CH) 2010-01-20 EP disclosed