SCHEMBL28755484

SCHEMBL28755484

CCC(=O)c1cc(Br)ccc1OC(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 3/20 0.42
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
ACHE P22303 1/20 0.40
HTR4 Q13639 1/20 0.40
ALPL P05186 3/20 0.39
F2R P25116 1/20 0.38
HMGCR P04035 1/20 0.37
EPHX2 P34913 1/20 0.37
KDR P35968 1/20 0.37
KCNK3 O14649 1/20 0.36
KCNK9 Q9NPC2 1/20 0.36
PPARG P37231 1/20 0.36
PTPN1 P18031 1/20 0.36
DDR1 Q08345 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3925476 0.86 MAOA (0.42) PTGDR2MAOAMAOBACHEHTR4
Hydrochloric Acid SCHEMBL30468019 0.84 MAOA (0.41) PTGDR2MAOAMAOBACHEHTR4
SCHEMBL30468068 0.83 PTGDR2 (0.56) PTGDR2MAOAMAOBALPLEPHX2
SCHEMBL15884099 0.83 PTGDR2 (0.56) PTGDR2MAOAMAOBALPLEPHX2
SCHEMBL937129 0.82 LMNA (0.47) PTGDR2
SCHEMBL29746555 0.82 KDM4E (0.50) PTGDR2MAOAMAOBALPLEPHX2
SCHEMBL2711853 0.82 KDM4E (0.50) PTGDR2MAOAMAOBALPLEPHX2
SCHEMBL28758200 0.82 ANO1 (0.45) ALPL
SCHEMBL15884087 0.82 NPSR1 (0.40) PTGDR2MAOAMAOBACHEALPL
SCHEMBL20855483 0.81 HMGCR (0.53) PTGDR2ACHEHTR4HMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100395234-C Novel CB1 receptor inverse agonists HOFFMANN LA ROCHE (CH) 2008-06-18 CN disclosed
CN-101012193-A Novel CB 1 receptour inverse agonists HOFFMANN LA ROCHE (CH) 2007-08-08 CN disclosed
CN-1735593-A Novel CB1 receptor inverse agonists HOFFMANN LA ROCHE (CH) 2006-02-15 CN disclosed