SCHEMBL28757336

SCHEMBL28757336

CCCCC1(F)Cc2ccccc2C1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX12 P18054 1/20 0.47
NPSR1 Q6W5P4 2/20 0.43
HTT P42858 2/20 0.43
LMNA P02545 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
POLB P06746 2/20 0.38
GAA P10253 2/20 0.37
KDM4E B2RXH2 1/20 0.37
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
HTR2A P28223 2/20 0.35
HTR2C P28335 2/20 0.35
HTR2B P41595 2/20 0.35
SIGMAR1 Q99720 2/20 0.35
ELANE P08246 1/20 0.35
CYP19A1 P11511 1/20 0.35
PRNP P04156 2/20 0.35
PPARG P37231 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
NR2E3 Q9Y5X4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12086639 0.79 ALOX12 (0.55) ALOX12NPSR1HTTLMNAL3MBTL1
SCHEMBL27973945 0.78 ALOX12 (0.47) ALOX12NPSR1HTTLMNAL3MBTL1
SCHEMBL25946601 0.77 ALOX12 (0.41) ALOX12SIGMAR1ALDH1A1CYP1A2CYP2C19
SCHEMBL12269439 0.76 NPSR1 (0.44) NPSR1HTTLMNAL3MBTL1POLB
SCHEMBL21882889 0.75 UTS2R (0.46) ALOX12NPSR1HTTLMNAL3MBTL1
SCHEMBL9342946 0.74 ALOX12 (0.49) ALOX12NPSR1HTTLMNAL3MBTL1
SCHEMBL12086597 0.72 GAA (0.49) ALOX12NPSR1HTTLMNAL3MBTL1
SCHEMBL29439376 0.72 NPSR1 (0.40) ALOX12NPSR1HTTLMNAL3MBTL1
SCHEMBL13253339 0.71 NPSR1 (0.57) ALOX12NPSR1HTTLMNAL3MBTL1
SCHEMBL27971438 0.71 NPSR1 (0.47) NPSR1HTTLMNAL3MBTL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102617464-A fused compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor ABBOTT LAB 2012-08-01 CN disclosed
CN-101445501-A Fused compounds that inhibit vanilloid receptor subtype 1 (VR1) receptor ABBOTT LAB (US) 2009-06-03 CN disclosed
CN-1835924-A Fused compounds that inhibit vanilloid receptor subtype 1(vr1) receptor ABBOTT LAB (US) 2006-09-20 CN disclosed