SCHEMBL28757397

SCHEMBL28757397

c1csc(CC[C](c2ncco2)c2ncco2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.41
CES1 P23141 4/20 0.40
FAAH O00519 1/20 0.40
NCEH1 Q6PIU2 1/20 0.40
TRPM8 Q7Z2W7 2/20 0.39
ADRA2A P08913 2/20 0.38
ADRA2B P18089 2/20 0.38
ADRA2C P18825 2/20 0.38
ME2 P23368 1/20 0.36
ME1 P48163 1/20 0.36
ME3 Q16798 1/20 0.36
POLB P06746 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
ADAM17 P78536 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
TSHR P16473 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27756446 0.74 NPC1 (0.38) CES1POLBSMN1; SMN2TSHRNPC1
SCHEMBL5458568 0.73 TAAR1 (0.46) TAAR1TRPM8ADRA2AADRA2BADRA2C
SCHEMBL27526772 0.69 RAB9A (0.43) CES1FAAHSMN1; SMN2NPC1RAB9A
SCHEMBL1309062 0.67
SCHEMBL7332254 0.66 TAAR1 (0.54) TAAR1ADRA2AADRA2BADRA2CPOLB
SCHEMBL10668826 0.66 TAAR1 (0.54) TAAR1TRPM8ADRA2AADRA2BADRA2C
SCHEMBL2030841 0.66 TAAR1 (0.71) TAAR1ADRA2AADRA2BADRA2CPOLB
SCHEMBL5759825 0.66 TRPM8 (0.39) TAAR1TRPM8POLBSMN1; SMN2NPC1
SCHEMBL654985 0.65 POLB (0.66) TAAR1ADRA2AADRA2BADRA2CPOLB
SCHEMBL6197785 0.65 TAAR1 (0.52) TAAR1ADRA2AADRA2BADRA2CPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1764651-A Quinazoline derivatives as antitumor agents ASTRAZENECA AB (SE) 2006-04-26 CN disclosed