SCHEMBL28757635

SCHEMBL28757635

NCc1ccc(CCn2c(N)nc3nc[nH]c3c2=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 6/20 0.47
ADORA3 P0DMS8 4/20 0.47
PNP P00491 2/20 0.41
MGMT P16455 1/20 0.40
NUDT1 P36639 2/20 0.38
CYP1A2 P05177 2/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
TOP2A P11388 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
CYP2C19 P33261 1/20 0.38
HIF1A Q16665 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CDK1 P06493 1/20 0.38
CCNB1 P14635 1/20 0.38
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38
CCNA1 P78396 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17186295 0.89 ADORA2B (0.46) ADORA2BADORA3PNPNUDT1CYP1A2
SCHEMBL18605503 0.89 ADORA3 (0.58) ADORA2BADORA3PNPMGMTNUDT1
SCHEMBL17186343 0.89 ADORA2B (0.49) ADORA2BADORA3PNPPDE4AADORA2A
SCHEMBL6268535 0.89 ADORA3 (0.60) ADORA2BADORA3PNPMGMTNUDT1
Hydrochloric Acid SCHEMBL18605473 0.88 ADORA2B (0.48) ADORA2BADORA3PNPPDE4AADORA2A
Hydrochloric Acid SCHEMBL17186530 0.88 ADORA3 (0.57) ADORA2BADORA3PNPMGMTNUDT1
Hydrochloric Acid SCHEMBL18605672 0.88 ADORA2B (0.46) ADORA2BADORA3PNPNUDT1CYP1A2
Hydrochloric Acid SCHEMBL17186430 0.88 ADORA3 (0.59) ADORA2BADORA3PNPMGMTNUDT1
SCHEMBL1262627 0.87 PNP (0.51) ADORA2BADORA3PNPMGMTPDE4A
SCHEMBL17186484 0.87 ADORA3 (0.53) ADORA2BADORA3PNPMGMTNUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1720332-A O6Substrates for -alkylguanine-DNA alkyltransferases ECOLE POLYTECH (CH) 2006-01-11 CN disclosed
CN-1717496-A Protein labelling with o6-alkylguanine-DNA alkyltransferase ECOLE POLYTECH (CH) 2006-01-04 CN disclosed