SCHEMBL28757702

SCHEMBL28757702

CC(C)(C)OC(=O)Nc1cc(-c2c[nH]nc2C(F)(F)F)ccn1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.40
AAK1 Q2M2I8 10/20 0.39
CYP3A4 P08684 3/20 0.39
PIK3C3 Q8NEB9 4/20 0.39
TGFBR1 P36897 1/20 0.39
GSK3B P49841 1/20 0.38
DYRK1A Q13627 1/20 0.38
IGF1R P08069 1/20 0.38
RIPK3 Q9Y572 1/20 0.38
UCHL1 P09936 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5360812 0.82 IRAK4 (0.44) IRAK4AAK1PIK3C3TGFBR1
SCHEMBL5354912 0.82 MAPK14 (0.47) IRAK4CYP3A4PIK3C3TGFBR1
SCHEMBL5353074 0.82 RIPK3 (0.45) GSK3BRIPK3
SCHEMBL5352411 0.80 GSK3B (0.45) IRAK4AAK1CYP3A4PIK3C3TGFBR1
SCHEMBL5349844 0.80 TGFBR1 (0.40) IRAK4AAK1PIK3C3TGFBR1GSK3B
SCHEMBL5355784 0.80 IRAK4 (0.42) IRAK4AAK1CYP3A4PIK3C3TGFBR1
SCHEMBL5349670 0.79 CDK9 (0.42) IRAK4AAK1PIK3C3TGFBR1GSK3B
SCHEMBL10129965 0.78 PIK3C3 (0.43) IRAK4AAK1CYP3A4PIK3C3TGFBR1
SCHEMBL1104982 0.75 RIPK3 (0.44) IRAK4AAK1PIK3C3TGFBR1GSK3B
SCHEMBL5251219 0.74 EGFR (0.57) IRAK4AAK1PIK3C3TGFBR1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100519552-C Pyrazole compounds UBE INDUSTRIES (JP) 2009-07-29 CN disclosed
CN-1684953-A Pyrazole compounds UBE INDUSTRIES (JP) 2005-10-19 CN disclosed