SCHEMBL28760130

SCHEMBL28760130

FC(F)(F)c1cccnc1N1CCN(c2cc(-c3cccc(Cl)c3)nc(CCBr)n2)CC1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 6/20 0.49
TRPA1 O75762 2/20 0.47
TRPV1 Q8NER1 2/20 0.42
CDK4 P11802 1/20 0.41
CCND3 P30281 1/20 0.41
GSK3B P49841 1/20 0.41
EPHX2 P34913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3877200 0.93 HSD11B1 (0.51) HSD11B1TRPA1TRPV1CDK4CCND3
SCHEMBL3880078 0.89 HSD11B1 (0.51) HSD11B1TRPA1TRPV1CDK4CCND3
SCHEMBL14613836 0.89 HSD11B1 (0.51) HSD11B1TRPA1TRPV1CDK4CCND3
SCHEMBL3878973 0.87 HSD11B1 (0.47) HSD11B1TRPA1TRPV1CDK4CCND3
SCHEMBL3879636 0.86 TRPV1 (0.49) HSD11B1TRPA1TRPV1CDK4CCND3
SCHEMBL13766131 0.85 HSD11B1 (0.47) HSD11B1TRPA1TRPV1CDK4CCND3
SCHEMBL3878966 0.84 HSD11B1 (0.48) HSD11B1TRPA1TRPV1CDK4CCND3
SCHEMBL3880711 0.84 HSD11B1 (0.45) HSD11B1TRPA1TRPV1CDK4CCND3
SCHEMBL3879429 0.84 HSD11B1 (0.53) HSD11B1TRPA1TRPV1EPHX2
SCHEMBL3879528 0.83 TRPA1 (0.51) HSD11B1TRPA1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1823057-A Biaryl piperazinyl-pyridine analogues NEUROGEN CORP (US) 2006-08-23 CN disclosed