SCHEMBL28763528

SCHEMBL28763528

O=C(O)c1cc2cc(CCO)ccc2[nH]1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMAD3 P84022 1/20 0.58
KDM4E B2RXH2 4/20 0.57
HPGD P15428 3/20 0.57
HSD17B10 Q99714 3/20 0.57
ALDH1A1 P00352 2/20 0.57
F7 P08709 1/20 0.57
F3 P13726 1/20 0.57
PIN1 Q13526 1/20 0.57
PDPK1 O15530 1/20 0.57
LMNA P02545 1/20 0.57
TSHR P16473 1/20 0.57
NFKB1 P19838 1/20 0.57
APEX1 P27695 1/20 0.57
CYP2C19 P33261 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
TBXAS1 P24557 1/20 0.54
PYGL P06737 2/20 0.53
SRD5A2 P31213 2/20 0.53
MAPT P10636 1/20 0.53
DAO P14920 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8360314 0.87 SMAD3 (0.62) SMAD3KDM4EHPGDHSD17B10ALDH1A1
SCHEMBL2421110 0.86 SMAD3 (0.57) SMAD3KDM4EHPGDHSD17B10ALDH1A1
SCHEMBL28474583 0.86 PIN1 (0.59) SMAD3KDM4EHPGDHSD17B10ALDH1A1
SCHEMBL6512147 0.86 SMAD3 (0.57) SMAD3KDM4EHPGDHSD17B10ALDH1A1
SCHEMBL28793315 0.86 KDM4E (0.59) SMAD3KDM4EHPGDHSD17B10ALDH1A1
SCHEMBL1144864 0.82 PIN1 (0.63) SMAD3KDM4EHPGDHSD17B10ALDH1A1
SCHEMBL6990262 0.82 SMAD3 (0.60) SMAD3KDM4EHPGDHSD17B10ALDH1A1
SCHEMBL5970277 0.82 KDM4E (0.63) SMAD3KDM4EHPGDHSD17B10ALDH1A1
SCHEMBL15642858 0.82 PLA2G4A (0.67) SMAD3KDM4EHPGDHSD17B10ALDH1A1
SCHEMBL27590744 0.82 SMAD3 (0.53) SMAD3KDM4EHPGDHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1972926-B Indole derivatives as histamine receptor antagonists HOFFMANN LA ROCHE 2011-02-16 CN disclosed
CN-1972926-A Indole derivatives as histamine receptor antagonists HOFFMANN LA ROCHE (CH) 2007-05-30 CN disclosed