SCHEMBL28768720

SCHEMBL28768720

C=CC(=O)N1CCN(C(=O)O)C(CO)C1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.39
TACR1 P25103 1/20 0.35
JAK3 P52333 5/20 0.34
TEAD1 P28347 6/20 0.33
POLB P06746 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TEAD3 Q99594 1/20 0.33
TET3 O43151 1/20 0.32
KMT2A Q03164 1/20 0.32
FBXL19 Q6PCT2 1/20 0.32
CXXC5 Q7LFL8 1/20 0.32
TET1 Q8NFU7 1/20 0.32
KDM2B Q8NHM5 1/20 0.32
CXXC4 Q9H2H0 1/20 0.32
KDM2A Q9Y2K7 1/20 0.32
BTK Q06187 5/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28768719 1.00 OPRK1 (0.39) OPRK1TACR1JAK3TEAD1POLB
SCHEMBL3766440 0.84 TACR1 (0.39) TACR1POLBL3MBTL1
SCHEMBL20744897 0.84 TACR1 (0.39) TACR1POLBL3MBTL1
SCHEMBL3766415 0.84 TACR1 (0.39) TACR1POLBL3MBTL1
SCHEMBL28880008 0.79 TACR1 (0.41) OPRK1TACR1POLBL3MBTL1
SCHEMBL24543498 0.78 NR1H2 (0.43) OPRK1
SCHEMBL28766609 0.78 NR1H2 (0.43) OPRK1
SCHEMBL22969760 0.78 OPRK1 (0.34) OPRK1JAK3TEAD1TEAD3BTK
SCHEMBL24543192 0.78 OPRK1 (0.34) OPRK1JAK3TEAD1TEAD3BTK
SCHEMBL20571063 0.76 TSHR (0.37) JAK3L3MBTL1TET3KMT2AFBXL19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114644631-A KRAS G12C protein mutation inhibitor, preparation method thereof, pharmaceutical composition and application thereof 上海维申医药有限公司 2022-06-21 CN disclosed