SCHEMBL28772995

SCHEMBL28772995

CC(=O)OC(c1ccccc1)(c1ccccc1)c1ccccc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 4/20 0.44
KCNA3 P22001 2/20 0.42
HTR2A P28223 2/20 0.41
HTR2C P28335 2/20 0.41
OPRK1 P41145 2/20 0.41
KCNH2 Q12809 2/20 0.41
ADRA1A P35348 1/20 0.41
KIF11 P52732 1/20 0.40
CYP1A2 P05177 3/20 0.38
KMT2A Q03164 3/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
CYP2C19 P33261 2/20 0.38
HIF1A Q16665 2/20 0.38
CYP2D6 P10635 2/20 0.38
MAPT P10636 2/20 0.38
MEN1 O00255 2/20 0.38
CYP3A4 P08684 2/20 0.38
TSHR P16473 2/20 0.38
GLA P06280 2/20 0.38
RAB9A P51151 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23110176 0.93 CYP2C9 (0.42) KCNN4KCNA3HTR2AHTR2COPRK1
SCHEMBL13940364 0.93 RAB9A (0.39) KCNN4KCNA3HTR2AHTR2COPRK1
SCHEMBL26348876 0.83 KIF11 (0.42) KIF11KMT2AMAPTMEN1CYP3A4
SCHEMBL20829082 0.83 KIF11 (0.42) KIF11KMT2AMAPTMEN1CYP3A4
SCHEMBL23110164 0.83 KIF11 (0.42) KIF11KMT2AMAPTMEN1CYP3A4
SCHEMBL5053673 0.83 KIF11 (0.45) KCNN4KCNA3HTR2AHTR2COPRK1
SCHEMBL1096837 0.82 KCNN4 (0.47) KCNN4KIF11CYP1A2KMT2ACYP2C19
SCHEMBL3401873 0.81 KCNN4 (0.38) KCNN4CYP1A2KMT2ACYP2C19HIF1A
SCHEMBL2406465 0.81 KCNN4 (0.42) KCNN4KCNA3HTR2AHTR2COPRK1
SCHEMBL28773038 0.80 KCNH2 (0.40) KCNN4KCNA3HTR2AHTR2COPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114729006-A Cyclic peptide compounds having Kras inhibitory activity 中外制药株式会社 2022-07-08 CN disclosed