SCHEMBL2877356

SCHEMBL2877356

COc1cccc(CN(C(C(=O)NO)C(C)C)S(=O)(=O)c2ccc(OCCCCl)cc2)c1

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 19/20 0.67
MMP9 P14780 17/20 0.67
MMP13 P45452 17/20 0.67
MMP8 P22894 16/20 0.67
MMP1 P03956 1/20 0.52
MMP3 P08254 1/20 0.52
MMP14 P50281 1/20 0.52
MMP16 P51512 1/20 0.52
ADAM17 P78536 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2877354 1.00 MMP2 (0.67) MMP2MMP9MMP13MMP8MMP1
SCHEMBL2876068 0.93 MMP2 (0.72) MMP2MMP9MMP13MMP8
SCHEMBL2876062 0.93 MMP2 (0.72) MMP2MMP9MMP13MMP8
SCHEMBL2855090 0.92 MMP2 (0.71) MMP2MMP9MMP13MMP8
SCHEMBL2855092 0.92 MMP2 (0.71) MMP2MMP9MMP13MMP8
SCHEMBL2860130 0.91 BMP1 (0.62) MMP2MMP9MMP13MMP8MMP1
SCHEMBL2860128 0.91 BMP1 (0.62) MMP2MMP9MMP13MMP8MMP1
SCHEMBL2873171 0.90 MMP2 (0.73) MMP2MMP9MMP13MMP8
SCHEMBL2873176 0.90 MMP2 (0.73) MMP2MMP9MMP13MMP8
SCHEMBL2857354 0.89 MMP2 (0.64) MMP2MMP9MMP13MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2085379-A1 Arylsulfonamido-substituted hydroxamic acid derivatives Novartis AG (CH) 2009-08-05 EP claimed
US-7138432-B1 Arylsulfonamido-substituted hydroxamic acid derivatives NOVARTIS AG (CH) 2006-11-21 US claimed
EP-1202961-A1 ARYLSULFONAMIDO-SUBSTITUTED HYDROXAMIC ACID DERIVATIVES Novartis AG (CH) 2002-05-08 EP claimed
WO-2001010827-A1 ARYLSULFONAMIDO-SUBSTITUTED HYDROXAMIC ACID DERIVATIVES NOVARTIS AG (CH) 2001-02-15 WO claimed
EP-1202961-B1 ARYLSULFONAMIDO-SUBSTITUTED HYDROXAMIC ACID DERIVATIVES NOVARTIS AG (CH) 2010-01-20 EP disclosed
EP-2085379-A1 Arylsulfonamido-substituted hydroxamic acid derivatives Novartis AG (CH) 2009-08-05 EP disclosed