SCHEMBL28776335

SCHEMBL28776335

O=[N+]([O-])c1cc(-c2csc(-c3cccnc3C(F)(F)F)n2)ccc1OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EIF4E P06730 13/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
RECQL P46063 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44
NFKB1 P19838 1/20 0.44
MAPK1 P28482 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
CYP19A1 P11511 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3590056 0.90 EIF4E (0.44) EIF4EMEN1KMT2ACYP19A1CYP11B1
SCHEMBL3580015 0.77 EIF4E (0.47) EIF4ELMNAMAPTRECQLMEN1
SCHEMBL28780443 0.75 CTSV (0.45) LMNAMEN1KMT2AALDH1A1POLB
SCHEMBL1446807 0.74 EIF4E (0.42) EIF4ECYP19A1CYP11B1CYP11B2
SCHEMBL3581595 0.73 POLB (0.47) NPC1RAB9ASMN1; SMN2MAPTPOLB
SCHEMBL1447240 0.72 POLB (0.46) NPC1RAB9AMAPTPOLBNFKB1
SCHEMBL2685823 0.72 CYP11B1 (0.63) NPC1RAB9ALMNAMEN1KMT2A
SCHEMBL3598965 0.72 MEN1 (0.49) EIF4ENPC1RAB9ASMN1; SMN2LMNA
SCHEMBL3581708 0.72 TUBB4A (0.41) NPC1RAB9AMEN1KMT2ACYP19A1
SCHEMBL27764455 0.71 POLB (0.39) NPC1RAB9AMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101454285-B Oxadiazole derivatives as comt inhibitors PORTELA & CA SA 2012-06-27 CN disclosed
CN-101454285-A Oxadiazole derivatives as comt inhibitors PORTELA & CA SA (PT) 2009-06-10 CN disclosed