SCHEMBL28779341

SCHEMBL28779341

NC(=O)c1ccc(OC(F)(F)F)cc1C1CCC(CCN2CCC(C(=O)c3ccc(F)cc3)CC2)CC1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.51
HTR2C P28335 5/20 0.45
HTR2A P28223 3/20 0.45
HTR7 P34969 3/20 0.45
HTR6 P50406 3/20 0.45
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CCR2 P41597 1/20 0.43
KDM2B Q8NHM5 1/20 0.42
MGLL Q99685 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28779340 1.00 HSD11B1 (0.51) HSD11B1HTR2CHTR2AHTR7HTR6
SCHEMBL27758318 0.87 HSD11B1 (0.48) HSD11B1HTR2CHTR2AHTR7HTR6
SCHEMBL27758316 0.87 HSD11B1 (0.48) HSD11B1HTR2CHTR2AHTR7HTR6
SCHEMBL229148 0.84 HTR2C (0.45) HTR2CHTR2AHTR7HTR6LMNA
SCHEMBL230362 0.84 HTR2C (0.52) HTR2CHTR2AHTR7HTR6
SCHEMBL27737546 0.84 HTR2C (0.52) HTR2CHTR2AHTR7HTR6
SCHEMBL228591 0.83 HTR2C (0.46) HTR2CHTR2AHTR7HTR6LMNA
SCHEMBL230298 0.82 HTR2C (0.45) HTR2CHTR2AHTR7HTR6LMNA
SCHEMBL227200 0.82 LMNA (0.46) HTR2CHTR2AHTR7HTR6LMNA
SCHEMBL229122 0.81 HTR2C (0.44) HTR2CHTR2AHTR7HTR6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101384581-B Benzoyl-piperidine derivatives as 5HT2/D3 modulators HOFFMANN LA ROCHE 2013-09-18 CN claimed
CN-101384581-A Benzoyl-piperidine derivatives as 5HT2/D3 modulators HOFFMANN LA ROCHE (CH) 2009-03-11 CN claimed
CN-101384581-B Benzoyl-piperidine derivatives as 5HT2/D3 modulators HOFFMANN LA ROCHE 2013-09-18 CN disclosed
CN-101384581-A Benzoyl-piperidine derivatives as 5HT2/D3 modulators HOFFMANN LA ROCHE (CH) 2009-03-11 CN disclosed