SCHEMBL2877955

SCHEMBL2877955

Cc1sc(Nc2ccc(Cl)cc2)nc1C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.55
RAB9A P51151 5/20 0.51
SMN1; SMN2 Q16637 4/20 0.51
POLB P06746 2/20 0.51
PTGDR2 Q9Y5Y4 5/20 0.51
KDM1A O60341 1/20 0.49
ALDH1A1 P00352 5/20 0.48
GAA P10253 4/20 0.48
NPC1 O15118 4/20 0.48
KMT2A Q03164 4/20 0.48
MAPT P10636 4/20 0.48
MEN1 O00255 3/20 0.48
KDM4E B2RXH2 2/20 0.45
P2RX3 P56373 2/20 0.45
CACNA1B Q00975 1/20 0.45
APBA1 Q02410 1/20 0.45
CASP3 P42574 1/20 0.45
SENP8 Q96LD8 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
SENP6 Q9GZR1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16586316 0.86 GAA (0.63) DHODHRAB9ASMN1; SMN2POLBPTGDR2
SCHEMBL5035180 0.82 DHODH (0.61) DHODHRAB9ASMN1; SMN2ALDH1A1GAA
SCHEMBL2878494 0.82 PTGDR2 (0.52) DHODHRAB9ASMN1; SMN2POLBPTGDR2
SCHEMBL2876767 0.81 PTGDR2 (0.51) DHODHRAB9ASMN1; SMN2POLBPTGDR2
SCHEMBL4923649 0.79 SMN1; SMN2 (0.59) DHODHRAB9ASMN1; SMN2POLBALDH1A1
SCHEMBL2878623 0.79 MAPT (0.44) DHODHRAB9ASMN1; SMN2ALDH1A1GAA
SCHEMBL788893 0.79 TRPC3 (0.61) RAB9ASMN1; SMN2ALDH1A1KMT2AMAPT
SCHEMBL2873347 0.78 ALDH1A1 (0.50) RAB9ASMN1; SMN2POLBALDH1A1GAA
SCHEMBL22053468 0.77 GAA (0.40) DHODHRAB9ASMN1; SMN2POLBALDH1A1
SCHEMBL19667972 0.77 NPC1 (0.40) RAB9APOLBALDH1A1GAANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010012793-A1 FUNGICIDE AMINOTHIAZOLE DERIVATIVES BAYER CROPSCIENCE SA (FR) 2010-02-04 WO disclosed
CN-100509808-C Novel thiazole derivates HOFFMANN LA ROCHE (CH) 2009-07-08 CN disclosed
US-7371751-B2 Thiazole derivatives HOFFMANN-LA ROCHE INC. (US) 2008-05-13 US disclosed
EP-1694673-B1 THIAZOLE DERIVATES HOFFMANN LA ROCHE (CH) 2008-01-16 EP disclosed
CN-1890236-A Novel thiazole derivates HOFFMANN LA ROCHE (CH) 2007-01-03 CN disclosed
EP-1694673-A1 NOVEL THIAZOLE DERIVATES F.HOFFMANN-LA ROCHE AG (CH) 2006-08-30 EP disclosed
US-20050153962-A1 Thiazole derivatives HOFFMANN-LA ROCHE INC. 2005-07-14 US disclosed
WO-2005058887-A1 NOVEL THIAZOLE DERIVATES F. HOFFMANN-LA ROCHE AG (CH) 2005-06-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050153962-A1 Thiazole derivatives CNR1, CNR2, GPR119 DHODH 2367/4885RAB9A 1847/4885SMN1; SMN2 3460/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.