SCHEMBL28784154

SCHEMBL28784154

COC(=O)N1CN=Cc2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX4 Q99571 7/20 0.53
ADORA3 P0DMS8 2/20 0.41
BCHE P06276 1/20 0.41
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM4E B2RXH2 1/20 0.35
ADORA1 P30542 1/20 0.34
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
SCN4A P35499 1/20 0.34
SCN5A Q14524 1/20 0.34
SCN9A Q15858 1/20 0.34
P2RX1 P51575 1/20 0.34
P2RX3 P56373 1/20 0.34
P2RX7 Q99572 1/20 0.34
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
NOTUM Q6P988 1/20 0.34
MYC P01106 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29843231 0.85 ADORA1 (0.43) P2RX4ADORA3BCHEMEN1KMT2A
SCHEMBL7020595 0.84 BCHE (0.44) P2RX4BCHEMEN1KMT2AMAPK1
SCHEMBL30081007 0.80 P2RX4 (0.40) P2RX4LMNATSHRMAPK1SCN4A
SCHEMBL7029078 0.80 P2RX4 (0.40) P2RX4LMNATSHRMAPK1SCN4A
SCHEMBL28222693 0.79 LMNA (0.39) P2RX4LMNATSHRMAPK1SCN4A
SCHEMBL28223433 0.79 LMNA (0.49) P2RX4BCHELMNATSHRMAPK1
SCHEMBL28222695 0.78 P2RX4 (0.52) P2RX4ADORA3MEN1KMT2AKDM4E
SCHEMBL28223435 0.78 P2RX4 (0.53) P2RX4ADORA3KMT2AMAPK1
SCHEMBL28860614 0.76 P2RX4 (0.49) P2RX4MEN1KMT2ALMNAMAPK1
SCHEMBL27822676 0.76 P2RX4 (0.51) P2RX4BCHEMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101580505-B Derivatives of pyrrolo[2,1-b]quinazoline natural products, preparation method and application thereof UNIV SHENYANG PHARMACEUTICAL 2014-09-10 CN disclosed
CN-101580505-A Derivatives of pyrrolo[2,1-b]quinazoline natural products, preparation method and application thereof UNIV SHENYANG PHARMACEUTICAL (CN) 2009-11-18 CN disclosed