SCHEMBL2878432

SCHEMBL2878432

COC(=O)Cc1c(-c2ccc(Cl)c(S(=O)(=O)NCCc3ccccc3OC(F)(F)F)c2)[nH]c2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MGAM O43451 1/20 0.45
MAPT P10636 5/20 0.44
TP53 P04637 1/20 0.41
EGFR P00533 2/20 0.40
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
ALOX5 P09917 1/20 0.37
CXCR2 P25025 1/20 0.37
TACR1 P25103 1/20 0.37
HSD17B13 Q7Z5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2873488 0.92 MGAM (0.47) MGAMMAPTTP53EGFRLMNA
SCHEMBL2873653 0.91 MAPT (0.51) MGAMMAPTTP53EGFRLMNA
SCHEMBL2878392 0.88 MGAM (0.45) MGAMMAPTTP53LMNAPOLB
SCHEMBL2876512 0.85 MAPT (0.51) MGAMMAPTTP53LMNAPOLB
SCHEMBL2878384 0.84 MAPT (0.48) MGAMMAPTTP53EGFRALOX5
SCHEMBL2878351 0.81 ALOX5 (0.55) MAPTTP53ALOX5
SCHEMBL2880985 0.81 ALOX5 (0.46) MAPTEGFRALOX5
SCHEMBL2878435 0.80 EGFR (0.39) MAPTEGFRLMNATACR1
SCHEMBL2873463 0.80 ACLY (0.51) MAPTTP53ALOX5
SCHEMBL2872499 0.79 MGAM (0.46) MGAMMAPTHSD17B13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2066628-B1 2-PHENYL-INDOLES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS SANOFI AVENTIS (FR) 2010-10-20 EP disclosed
US-20090176804-A1 2-PHENYL-INDOLES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS SANOFI-AVENTIS (FR) 2009-07-09 US disclosed
EP-2066628-A1 2-PHENYL-INDOLES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS Sanofi-Aventis (FR) 2009-06-10 EP disclosed
WO-2008014186-A1 2-PHENYL-INDOLES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS SANOFI-AVENTIS (FR) 2008-01-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090176804-A1 2-PHENYL-INDOLES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS PTGER2, PTGDR2, CYSLTR2 MGAM 4301/4885MAPT 2271/4885TP53 3735/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.