SCHEMBL28784608

SCHEMBL28784608

FC(F)(F)c1cccc(-c2cc(CCBr)no2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
RAB9A P51151 4/20 0.43
GAA P10253 1/20 0.43
MAPK1 P28482 1/20 0.43
BRD4 O60885 1/20 0.43
NPC1 O15118 2/20 0.42
POLB P06746 2/20 0.42
MAPT P10636 2/20 0.42
CXCR1 P25024 1/20 0.41
NOTUM Q6P988 2/20 0.41
S1PR1 P21453 2/20 0.41
EPHX2 P34913 1/20 0.40
CASP3 P42574 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2109752 0.89 RAB9A (0.45) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL28946942 0.84 SIRT2 (0.48) CYP3A4CYP2C19RAB9APOLBMAPT
SCHEMBL2428467 0.83 RAB9A (0.45) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL2107054 0.83 NOTUM (0.62) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL12444310 0.83 BRD4 (0.48) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5559631 0.80 POLB (0.46) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL27163705 0.79 NOTUM (0.64) CYP1A2CYP2D6CYP2C9CYP2C19RAB9A
SCHEMBL27591767 0.78 RAB9A (0.48) RAB9AMAPK1NPC1POLBMAPT
SCHEMBL3630996 0.75 BRD4 (0.55) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL11256348 0.75 BRD4 (0.55) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101925590-A Aldh-2 inhibitors in treatment of addiction CV THERAPEUTICS INC 2010-12-22 CN disclosed
CN-101627024-A ALDH-2 inhibitors in the treatment of addiction CV THERAPEUTICS INC 2010-01-13 CN disclosed