SCHEMBL2878614

SCHEMBL2878614

Fc1cnc(Cl)nc1-c1cc2cccc(-c3ccncc3CN3CCOCC3)c2s1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 5/20 0.37
JAK1 P23458 4/20 0.37
TYK2 P29597 4/20 0.37
JAK3 P52333 4/20 0.37
IKBKE Q14164 1/20 0.36
TBK1 Q9UHD2 1/20 0.36
MCHR1 Q99705 1/20 0.35
CYP2A13 Q16696 3/20 0.35
KCNH2 Q12809 1/20 0.35
AURKA O14965 1/20 0.35
AURKB Q96GD4 1/20 0.35
TGFBR1 P36897 1/20 0.34
TGFBR2 P37173 1/20 0.34
METAP2 P50579 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
PAX8 Q06710 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
RPS6KA3 P51812 1/20 0.34
ADORA2A P29274 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2875961 0.89 JAK2 (0.38) JAK2JAK1TYK2JAK3MCHR1
SCHEMBL27776237 0.87 ADORA2A (0.38) JAK2JAK1TYK2JAK3MCHR1
SCHEMBL1339059 0.81 ADORA2A (0.35) JAK2JAK1TYK2JAK3KCNH2
SCHEMBL1336736 0.78 JAK2 (0.36) JAK2JAK1TYK2JAK3MCHR1
SCHEMBL394127 0.77 LIMK1 (0.31) RPS6KA3
SCHEMBL388969 0.75 PIP4K2A (0.33)
SCHEMBL391723 0.75 ALDH1A1 (0.37) METAP2RPS6KA3GSK3B
SCHEMBL2923179 0.75 TDO2 (0.39) ADORA2AADORA1GSK3B
SCHEMBL391679 0.74 ALDH1A1 (0.31)
SCHEMBL2879097 0.73 CXCR4 (0.41) CYP2A13ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125794-B1 IMIDAZOLIDINONYL AMINOPYRIMIDINE COMPOUNDS FOR THE TREATMENT OF CANCER LILLY CO ELI (US) 2010-10-20 EP disclosed