SCHEMBL28790263

SCHEMBL28790263

O=C(O)Cc1nc(Br)sc1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
MAPT P10636 1/20 0.45
KDM4E B2RXH2 3/20 0.44
GRK6 P43250 1/20 0.44
ADORA1 P30542 1/20 0.44
KMO O15229 2/20 0.43
RORB Q92753 1/20 0.43
RXRA P19793 2/20 0.43
RXRB P28702 2/20 0.43
RXRG P48443 2/20 0.43
CTSK P43235 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
ALPL P05186 1/20 0.42
ALPI P09923 1/20 0.42
XDH P47989 1/20 0.42
PIN1 Q13526 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27837167 0.86 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL27803420 0.86 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL27803395 0.83 KDM4E (0.53) ALDH1A1SMN1; SMN2KDM4EPTGDR2
SCHEMBL27818022 0.82 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL27803413 0.81 KDM4E (0.56) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL27803404 0.81 KDM4E (0.46) ALDH1A1SMN1; SMN2KMT2AMAPTKDM4E
SCHEMBL2994499 0.81 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL27803418 0.79 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL28790262 0.77 ALOX5 (0.49) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL27803416 0.74 KDM4E (0.50) ALDH1A1KDM4EPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102164896-A Phenethylamide derivatives and their heterocyclic analogues ACTELION PHARMACEUTICALS LTD 2011-08-24 CN disclosed
CN-101965343-A 2-aza-bicyclo[2.2.1]heptane derivatives ACTELION PHARMACEUTICALS LTD 2011-02-02 CN disclosed