SCHEMBL28790705

SCHEMBL28790705

Brc1ccc([C@@H]2C=Cc3ccccc3O2)cc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
NPC1 O15118 1/20 0.33
GAA P10253 1/20 0.33
HDAC4 P56524 1/20 0.33
AHR P35869 1/20 0.32
TP53 P04637 5/20 0.31
MDM2 Q00987 5/20 0.31
NR3C1 P04150 1/20 0.31
PGR P06401 1/20 0.31
NR3C2 P08235 1/20 0.31
AR P10275 1/20 0.31
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25190010 1.00 MEN1 (0.39) MEN1KMT2ANFKB1NFKB2RELA
SCHEMBL25264499 1.00 MEN1 (0.39) MEN1KMT2ANFKB1NFKB2RELA
SCHEMBL17227883 0.85 NFKB1 (0.38) MEN1KMT2ANFKB1NFKB2RELA
SCHEMBL17229229 0.85 NFKB1 (0.38) MEN1KMT2ANFKB1NFKB2RELA
SCHEMBL725410 0.85 NFKB1 (0.38) MEN1KMT2ANFKB1NFKB2RELA
SCHEMBL30315348 0.85 NFKB1 (0.38) MEN1KMT2ANFKB1NFKB2RELA
SCHEMBL17227902 0.84 MAOB (0.40) MEN1KMT2ANFKB1NFKB2RELA
SCHEMBL25201323 0.84 MAOB (0.40) MEN1KMT2ANFKB1NFKB2RELA
SCHEMBL15954244 0.84 MAOB (0.40) MEN1KMT2ANFKB1NFKB2RELA
SCHEMBL25193070 0.83 POLB (0.39) MEN1KMT2ANFKB1NFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101921252-B 1-oxa-benzo-heterocycle compound, synthesis method and application thereof SHANGHAI INST ORGANIC CHEM 2012-05-09 CN disclosed
CN-101921252-A 1-oxa-benzo-heterocycle compound, synthesis method and application thereof SHANGHAI INST ORGANIC CHEM 2010-12-22 CN disclosed