SCHEMBL28790992

SCHEMBL28790992

CC(CO)NC(=O)c1cc(-c2ccc(Cl)cn2)cc(-n2ncnc2C(F)(F)F)c1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 11/20 0.48
P2RX2 Q9UBL9 10/20 0.48
CYP2C9 P11712 1/20 0.44
HDAC4 P56524 1/20 0.44
MAP4K4 O95819 1/20 0.43
AHR P35869 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2278031 1.00 P2RX3 (0.48) P2RX3P2RX2CYP2C9HDAC4MAP4K4
SCHEMBL2273906 0.94 P2RX3 (0.48) P2RX3P2RX2CYP2C9HDAC4MAP4K4
SCHEMBL2277313 0.92 P2RX3 (0.49) P2RX3P2RX2CYP2C9MAP4K4AHR
SCHEMBL27830176 0.90 P2RX3 (0.59) P2RX3P2RX2
SCHEMBL2272068 0.90 P2RX3 (0.59) P2RX3P2RX2
SCHEMBL2273162 0.89 P2RX3 (0.49) P2RX3P2RX2MAP4K4AHR
SCHEMBL4318767 0.89 P2RX3 (0.46) P2RX3P2RX2CYP2C9HDAC4MAP4K4
SCHEMBL27748147 0.89 P2RX3 (0.46) P2RX3P2RX2CYP2C9HDAC4MAP4K4
SCHEMBL2272715 0.89 P2RX3 (0.47) P2RX3P2RX2MAP4K4AHR
SCHEMBL2272521 0.89 P2RX3 (0.47) P2RX3P2RX2MAP4K4AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101903359-A Triazole-substituted arylamide derivatives and their use as P2X3And/or P2X2/3Use of purinergic receptor antagonists HOFFMANN LA ROCHE 2010-12-01 CN disclosed