SCHEMBL28792255

SCHEMBL28792255

COc1cc(O)c2occc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.47
MAOA P21397 3/20 0.42
MAPK1 P28482 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2A6 P11509 1/20 0.42
TSHR P16473 1/20 0.42
ACHE P22303 1/20 0.42
PDE4A P27815 1/20 0.42
CYP2C19 P33261 1/20 0.42
SLC6A3 Q01959 1/20 0.42
CYP2A13 Q16696 1/20 0.42
ABL1 P00519 6/20 0.42
BCR P11274 6/20 0.42
ABCB1 P08183 5/20 0.42
CYP1A1 P04798 4/20 0.42
CYP1B1 Q16678 4/20 0.42
ALOX5 P09917 3/20 0.42
PTGS2 P35354 3/20 0.42
KDM4E B2RXH2 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5689313 0.85 ALOX5 (0.58) CYP3A4MAPK1CYP1A2ABL1BCR
SCHEMBL5689322 0.85 ALOX5 (0.58) CYP3A4MAPK1CYP1A2ABL1BCR
SCHEMBL5689317 0.85 ALOX5 (0.58) CYP3A4MAPK1CYP1A2ABL1BCR
SCHEMBL10044955 0.81 CYP3A4 (0.42) CYP3A4MAOAMAPK1CYP1A2CYP2D6
SCHEMBL4984623 0.81 MAOA (0.42) CYP3A4MAOAMAPK1CYP1A2CYP2D6
SCHEMBL119906 0.81 CYP3A4 (0.47) CYP3A4MAOAMAPK1CYP1A2CYP2D6
SCHEMBL19783319 0.79 CYP1A2 (0.41) CYP3A4MAOAMAPK1CYP1A2CYP2D6
SCHEMBL4295622 0.79 MAOA (0.48) CYP3A4MAOAMAPK1CYP1A2CYP2D6
SCHEMBL7483039 0.79 MKNK2 (0.43) CYP1A2CYP2A6CYP1A1CYP1B1ALOX5
SCHEMBL9097330 0.78 CDC25B (0.48) CYP3A4MAOAMAPK1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114761410-B Pyrrolopyrimidinone compounds and application thereof 广州必贝特医药股份有限公司 2023-08-25 CN disclosed
WO-2022213932-A1 PYRROLOPYRIMIDINONE COMPOUND AND APPLICATION THEREOF 广州必贝特医药股份有限公司 2022-10-13 WO disclosed
CN-114761410-A Pyrrolopyrimidinone compounds and application thereof 广州必贝特医药股份有限公司 2022-07-15 CN disclosed