SCHEMBL28792500

SCHEMBL28792500

COc1c(Br)c(-c2ccccc2)c(C=O)c(OC)c1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 7/20 0.42
PDE4A P27815 5/20 0.42
PDE4C Q08493 5/20 0.42
PDE4D Q08499 5/20 0.42
ALDH1A1 P00352 2/20 0.38
LCK P06239 1/20 0.38
GLA P06280 1/20 0.38
MAPT P10636 1/20 0.38
THRB P10828 1/20 0.38
LIMK1 P53667 1/20 0.38
LIMK2 P53671 1/20 0.38
MGAM O43451 1/20 0.37
GAA P10253 1/20 0.37
SI P14410 1/20 0.37
MGAM2 Q2M2H8 1/20 0.37
RAB9A P51151 1/20 0.35
ERN1 O75460 2/20 0.35
AR P10275 1/20 0.34
MCL1 Q07820 1/20 0.33
CA1 P00915 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28339601 0.86 PDE4B (0.47) PDE4BPDE4APDE4CPDE4DALDH1A1
SCHEMBL29672050 0.83 PDE4B (0.50) PDE4BPDE4APDE4CPDE4DALDH1A1
SCHEMBL24049430 0.77 MGAM (0.56) PDE4BPDE4APDE4CPDE4DALDH1A1
SCHEMBL8684241 0.74 PTPN1 (0.41) ALDH1A1LCKGLAMAPTTHRB
SCHEMBL21384700 0.73 PDE4B (0.55) PDE4BPDE4APDE4CPDE4DALDH1A1
SCHEMBL21661958 0.71 LMNA (0.41) ALDH1A1MAPTTHRBGAARAB9A
SCHEMBL29672046 0.71 PDE4B (0.54) PDE4BPDE4APDE4CPDE4DALDH1A1
SCHEMBL16056248 0.71 PDE4B (0.42) PDE4BPDE4APDE4CPDE4DALDH1A1
SCHEMBL21661959 0.70 AR (0.40) ALDH1A1MAPTRAB9AAR
SCHEMBL25742898 0.69 MGAM (0.49) PDE4BPDE4APDE4CPDE4DALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112961041-B Catechol compound and preparation method and application thereof 心远(广州)药物研究有限公司 2022-06-21 CN disclosed
CN-112961041-A Catechol compound and preparation method and application thereof 心远(广州)药物研究有限公司 2021-06-15 CN disclosed