SCHEMBL8684241

SCHEMBL8684241

COc1c(Br)c(C=O)c(OC)c(OC)c1OC

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.41
ERN1 O75460 3/20 0.40
CA2 P00918 4/20 0.38
CA4 P22748 3/20 0.38
CA1 P00915 2/20 0.38
CA6 P23280 1/20 0.38
PRKDC P78527 1/20 0.38
AKR1B1 P15121 2/20 0.33
ALDH1A1 P00352 2/20 0.31
LCK P06239 1/20 0.30
GLA P06280 1/20 0.30
MAPT P10636 1/20 0.30
THRB P10828 1/20 0.30
LIMK1 P53667 1/20 0.30
LIMK2 P53671 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15961260 0.88 PTPN1 (0.48) PTPN1ERN1CA2CA4CA1
SCHEMBL18270044 0.83 ERN1 (0.41) PTPN1ERN1CA2CA4CA1
SCHEMBL5082572 0.82 AKR1B1 (0.38) ERN1CA2CA1PRKDCAKR1B1
SCHEMBL28363113 0.79 AKR1B1 (0.37) ERN1CA2CA1PRKDCAKR1B1
SCHEMBL10503320 0.76 ERN1 (0.49) PTPN1ERN1CA2CA1PRKDC
SCHEMBL3749542 0.76 ALDH1A1 (0.50) ERN1CA2CA1PRKDCALDH1A1
SCHEMBL28792500 0.74 PDE4B (0.42) ERN1CA2CA1ALDH1A1LCK
SCHEMBL6922829 0.74 ERN1 (0.39) PTPN1ERN1CA2CA4CA1
SCHEMBL19021119 0.74 SMN1; SMN2 (0.39) PTPN1ERN1CA2CA4CA1
SCHEMBL4264149 0.74 CA2 (0.52) ERN1CA2CA4CA1CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731455-A ALKYL 2-ALKYLACYLACRYLATE CHEMICAL INTERMEDIATE; ANTICHOLESTEROL AGENTS SHIONOGI & CO., LTD. (JP) 1998-03-24 US disclosed
EP-0597107-B1 LIGNAN ANALOG, PRODUCTION THEREOF, AND HYPOLIPIDEMIC DRUG SHIONOGI & CO (JP) 1996-07-03 EP disclosed
US-5502216-A ANTICHOLESTEROL SHIONOGI & CO., LTD. (JP) 1996-03-26 US disclosed
EP-0701991-A1 Process for the preparation of lignin analogues and starting materials therefor SHIONOGI & CO., LTD. (JP) 1996-03-20 EP disclosed
US-5449814-A Dehydration; Michael condensation SHIONOGI & CO., LTD. (JP) 1995-09-12 US disclosed
US-5420333-A Hydroxy ketone compounds SHIONOGI & CO., LTD. (JP) 1995-05-30 US disclosed
EP-0597107-A1 LIGNAN ANALOG, PRODUCTION THEREOF, AND HYPOLIPIDEMIC DRUG SHIONOGI & CO., LTD. (JP) 1994-05-18 EP disclosed