SCHEMBL28794894

SCHEMBL28794894

COc1cccc(-n2c(C)c(C#N)c3ccc(Br)cc32)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.43
MAPT P10636 4/20 0.43
LMNA P02545 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 2/20 0.43
PABPC1 P11940 1/20 0.43
MAPK1 P28482 1/20 0.43
CASP3 P42574 1/20 0.43
NCOA1 Q15788 1/20 0.43
SENP6 Q9GZR1 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
NCOA3 Q9Y6Q9 1/20 0.43
GAA P10253 2/20 0.40
NOTUM Q6P988 1/20 0.39
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
TDP2 O95551 1/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10192294 0.88 CLK1 (0.43) HTTMAPTLMNAMEN1KMT2A
SCHEMBL4066328 0.82 HTT (0.56) HTTMAPTLMNAMEN1KMT2A
SCHEMBL25946273 0.74 EGFR (0.38) HTTMAPTLMNAMEN1KMT2A
SCHEMBL346299 0.73 TSPO (0.49) HTTMAPTMEN1KMT2AKDM4E
SCHEMBL4066605 0.72 CLK1 (0.60) HTTMAPTLMNAMEN1KMT2A
SCHEMBL10095267 0.72 EDNRA (0.48) HTTMAPTLMNAMEN1KMT2A
SCHEMBL4794811 0.71 CLK1 (0.53) HTTMAPTLMNAMEN1KMT2A
SCHEMBL10134266 0.71 KDM4E (0.46) HTTMAPTLMNAMEN1KMT2A
SCHEMBL5577123 0.71 KDM4E (0.44) HTTMAPTLMNAMEN1KMT2A
SCHEMBL4056293 0.70 CLK1 (0.43) HTTMAPTLMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102020601-B Method for synthesizing N-aryl indole-3-nitrile derivative UNIV TIANJIN 2012-10-24 CN disclosed
CN-102020601-A Method for synthesizing N-aryl indole-3-nitrile derivative UNIV TIANJIN 2011-04-20 CN disclosed