SCHEMBL28795283

SCHEMBL28795283

CC(Br)c1cccc(OC(F)(F)F)c1[N+](=O)[O-]

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 3/20 0.40
KCNK9 Q9NPC2 3/20 0.40
P2RX7 Q99572 1/20 0.39
ALDH1A1 P00352 4/20 0.36
TDP1 Q9NUW8 2/20 0.36
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
TP53 P04637 2/20 0.33
TSHR P16473 1/20 0.33
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
MAPT P10636 2/20 0.32
MEN1 O00255 1/20 0.32
CASP3 P42574 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
SENP7 Q9BQF6 1/20 0.32
EPAS1 Q99814 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16956170 0.87 KCNK3 (0.39) KCNK3KCNK9ALDH1A1TDP1AKR1C3
SCHEMBL16951764 0.80 KCNK3 (0.33) KCNK3KCNK9ALDH1A1TDP1AKR1C3
SCHEMBL16958356 0.78 ALDH1A1 (0.58) ALDH1A1TDP1AKR1C3AKR1C2TP53
SCHEMBL26922160 0.78 AKR1C3 (0.36) ALDH1A1TDP1AKR1C3AKR1C2TP53
SCHEMBL16954493 0.78 KCNK3 (0.34) KCNK3KCNK9AKR1C3AKR1C2TP53
SCHEMBL3779733 0.78 NPC1 (0.36) KCNK3KCNK9ALDH1A1TDP1AKR1C3
SCHEMBL27703298 0.77 KCNK3 (0.43) KCNK3KCNK9P2RX7ALDH1A1PDE9A
SCHEMBL28798122 0.77 P2RX7 (0.57) P2RX7ALDH1A1TDP1AKR1C3AKR1C2
SCHEMBL10524671 0.76 MAPT (0.40) ALDH1A1TDP1AKR1C3AKR1C2TP53
SCHEMBL30806803 0.76 P2RX7 (0.44) KCNK3KCNK9P2RX7ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102482221-A Bicyclic and tricyclic compounds as KATII inhibitors PFIZER 2012-05-30 CN disclosed